Target Details
UniProt ACP37288
Gene SymbolAVPR1A
Protein NameVasopressin V1a receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1) PF08983 (V1R_C)
Summary
  • Multi-target molecules 537
  • Clinical molecules 0
  • Avg pChEMBL 7.48
Top Co-occurrence Targets
Active Molecules (537)
InChIKey pChEMBL Type Targets Clinical
NBCJMCYBNVOOFP 6.4 IC50 2
NBLUMDFJQQALBR 6.4 Ki 3
JTBHLQXMGZKKRH 6.4 Ki 2
KSNUCNRMDYJBKT 6.4 IC50 3
GBSJGFNEBBZCKT 6.4 IC50 3
RTYFXNURHRXECA 6.4 Ki 2
YUZYROBUIAUGNA 6.4 IC50 3
IBRRMWAYJVCIAO 6.4 Ki 2
DRCJSVOKCHFWFD 6.4 IC50 2
DGNLGAPGUAAZJA 6.4 Ki 2
NGYIKLFRMYALTL 6.4 IC50 2
NYBROGHBIFFJKW 6.4 Ki 3
NYBROGHBIFFJKW 6.4 Ki 3
SFPMVILWAAMPNK 6.3 Ki 2
JXKQHDZUZGKDGO 6.3 Ki 3
TYMAZOPJSZRWRR 6.3 Ki 2
TYMAZOPJSZRWRR 6.3 Ki 2
HZOABPDJUQEYFK 6.3 IC50 2
AQDLQNVRLVJCSR 6.3 IC50 3
IAGBXLVADMVFOS 6.3 Ki 2
TUPGNQOJPVCCLD 6.3 IC50 2
YPEFEMMVRUXHMR 6.3 Ki 2
XSVCEDLKELNLBS 6.3 Ki 3
ZYPZICFGURDSJH 6.3 Ki 2
DJBBIRTUOREGET 6.3 Ki 3
JDYXUSPYOGWCEU 6.3 Ki 2
JMGDUUQAXVYNKR 6.3 Ki 2
QIEUMSLIZIBCSF 6.3 Ki 3
ZJWAEMNLDJQLSS 6.3 Ki 3
AGEXZVIELPYYMU 6.3 IC50 2
YNHNTIWPKSQSOZ 6.3 IC50 2
BPRTVWSFENDHFX 6.3 Ki 2
WRHPPQZOFSXDOM 6.3 Ki 2
TUHHRVOIMGMMSL 6.2 Ki 2
BSYIUTMEBAJKRA 6.2 IC50 2
CMWAFGVDYAWHSS 6.2 Ki 2
KBCWEFINRBPCKH 6.2 Ki 2
ZJPXAVVKRGAFRV 6.2 Ki 3
PEQYLPNRGBWXGI 6.2 Ki 2
MIWKBPHMEDNABW 6.2 IC50 2
YCUKNIRQPJXXQQ 6.2 Ki 2
CZRITFDAPBAXMY 6.2 Ki 3
JLDUHYJPNRGFMT 6.2 Ki 3
KADSBHRUZZTVJC 6.2 Ki 2
KUYYTTWJIWYFTJ 6.2 Ki 3
XVTJVQICSDHKDD 6.2 Ki 2
DPJXIUXSMVOLCY 6.2 IC50 2
TYWBAYRNYLDJBB 6.2 Ki 2
YDQFMQKHNPCEQF 6.2 Ki 2
BIZKRBBLYHMLOO 6.2 Ki 2
2D structure