Target Details
UniProt ACP37288
Gene SymbolAVPR1A
Protein NameVasopressin V1a receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1) PF08983 (V1R_C)
Summary
  • Multi-target molecules 537
  • Clinical molecules 0
  • Avg pChEMBL 7.48
Top Co-occurrence Targets
Active Molecules (537)
InChIKey pChEMBL Type Targets Clinical
SDDPQRKDOGENES 10.3 Ki 2
HHUHDROQLLILRW 10.2 Ki 2
SDDBZVPPXOIBKA 10.1 Ki 4
PWTMAMJBZUGMBO 10.1 Ki 3
SVLGRIWNJNOFJU 10.1 Ki 3
BRYITMVYUBPGDS 10.0 Ki 2
SXYAVSQTBRVYRE 9.8 Ki 3
ANLGSZHSYWTWCO 9.6 Ki 2
VDUUABBYYOPFAW 9.5 Ki 3
SCNLVBYDEIZTGQ 9.5 Ki 2
DZTLOLIBSNAFTP 9.4 Ki 2
KHQMNMAJGZDPLL 9.3 IC50 2
LWIFUMBSEFSLJP 9.3 IC50 2
LFXCGLFTXRJJLT 9.3 IC50 3
UJXPNHJXBUDOGG 9.3 Ki 2
NKXUAADXAUNSRR 9.2 IC50 2
NKXUAADXAUNSRR 9.2 IC50 2
ICRPTZMWRJGNQI 9.2 Ki 2
VWXRQYYUEIYXCZ 9.2 Ki 4
JPBNIWAIRSKBSQ 9.2 Ki 2
UWSDXHIYRAYHRD 9.2 Ki 4
CSGBQCRJBAYXNV 9.1 IC50 2
NKXUAADXAUNSRR 9.1 IC50 2
CEBYCSRFKCEUSW 9.1 Ki 2
GEBXIWZNCWWKDS 9.1 Ki 2
XPJLLCAORNNZCL 9.1 Ki 2
ZENOFYULYVVPCE 9.1 Ki 4
PECYYLGJQLWWIB 9.1 IC50 2
QDPVGLNUJIYJDL 9.0 Ki 2
VTNGPTMGAMBQQJ 9.0 IC50 2
WEFIJLZIAONNPW 9.0 IC50 2
LZBBZUWWQMKLNP 9.0 Ki 2
KYIGOCCCBXRHNJ 9.0 IC50 43
IKENVDNFQMCRTR 8.9 IC50 2
XBYRXDQUZUKNHF 8.9 IC50 2
PECYYLGJQLWWIB 8.9 IC50 2
HKNSUPCHOJIVAF 8.9 IC50 2
KBZOIRJILGZLEJ 8.9 Ki 4
PICUPEIXWHWVFR 8.9 IC50 2
GDIIZZKPPFKLLK 8.9 IC50 2
WTDORPHQLSCAEW 8.9 IC50 2
VFXPCVBUMMROTO 8.9 IC50 2
IMYGSCWUXRQNTN 8.8 IC50 2
DCYBXBMLQQZOBV 8.8 Ki 4
DCYBXBMLQQZOBV 8.8 Ki 4
IMYGSCWUXRQNTN 8.8 IC50 2
KOVUSQJAPVOSKT 8.8 IC50 2
QDPVGLNUJIYJDL 8.8 Ki 2
YLKRSDQVBIBIIN 8.8 IC50 2
RPDVXKRTSHQHKP 8.8 IC50 2
2D structure