Target Details
| UniProt AC | P37173 |
|---|---|
| Gene Symbol | TGFBR2 |
| Protein Name | TGF-beta receptor type-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08917 (ecTbetaR2) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 144
- Clinical molecules 7
- Avg pChEMBL 6.66
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
- Transcriptional misregulation in cancer
Associated Diseases (6)
Active Molecules (144)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RIAWKODQFUGNFD
|
6.2 | IC50 | 2 | — | |
BYPWTZRGWLOOAC
|
6.2 | IC50 | 2 | — | |
SLMLHNHQKOPWPC
|
6.2 | IC50 | 2 | — | |
SXNCFFITOIFUMU
|
6.2 | IC50 | 2 | — | |
KYGGBIHPYVWDIQ
|
6.2 | IC50 | 2 | — | |
DEBKOHRICHTOCP
|
6.2 | IC50 | 2 | — | |
FFEWOBPMLFVMPC
|
6.2 | IC50 | 2 | — | |
IPESYYFOXATSFJ
|
6.2 | IC50 | 3 | — | |
ORRRLMFZEDPMSZ
|
6.2 | IC50 | 2 | — | |
QLCHJBPDLYRMBA
|
6.2 | IC50 | 2 | — | |
JMGXJHWTVBGOKG
|
6.2 | Kd | 7 | — | |
UARVSLPFGRKWQN
|
6.2 | IC50 | 11 | — | |
DGTYEYRETGUTQA
|
6.1 | IC50 | 2 | — | |
XPASUDUUTHMDBC
|
6.1 | IC50 | 2 | — | |
WTZAWAYSHRQGOB
|
6.1 | IC50 | 2 | — | |
XGEBOBAOVSOQCV
|
6.1 | IC50 | 10 | — | |
XNECSXXXAVERCS
|
6.1 | IC50 | 2 | — | |
OMZCMEYTWSXEPZ
|
6.1 | Kd | 43 | Yes | |
WOKGXNSTAOLINW
|
6.1 | IC50 | 2 | — | |
BTEPRNNLWBMDPC
|
6.1 | IC50 | 2 | — | |
HUEXJRRSSHIGFJ
|
6.1 | IC50 | 2 | — | |
IRFYJXPFDRTUSQ
|
6.1 | IC50 | 2 | — | |
WWTRFWLRGARRAD
|
6.1 | IC50 | 10 | — | |
XQRVINZFDOUPSD
|
6.1 | IC50 | 2 | — | |
XTCDENUICFWZKD
|
6.1 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
6.1 | Kd | 200 | — | |
CSZAJEXPQFERTK
|
6.1 | IC50 | 10 | — | |
LILHDFQTAZTSON
|
6.1 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
6.1 | Kd | 64 | Yes | |
NZEXAUMJUOFREM
|
6.0 | IC50 | 2 | — | |
YZDJQTHVDDOVHR
|
6.0 | Kd | 23 | — | |
XNVAPQIDSALKTN
|
6.0 | IC50 | 2 | — | |
HCZOMSNBQCWQJO
|
6.0 | IC50 | 2 | — | |
MGPDWDBEWFYGJF
|
6.0 | IC50 | 2 | — | |
OASUZJWWTNKKNW
|
6.0 | IC50 | 2 | — | |
BLZGGHVIKCCXDY
|
6.0 | IC50 | 2 | — | |
CPUGCQQDYFHDEM
|
6.0 | IC50 | 2 | — | |
STPUEPLVTCNYHC
|
6.0 | IC50 | 2 | — | |
JFQUUTOBSZUMCQ
|
6.0 | IC50 | 2 | — | |
HJZCMIKTRDMVQA
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
SXDZOHOHBPOZQD
|
6.0 | IC50 | 2 | — |