Target Details
| UniProt AC | P37173 |
|---|---|
| Gene Symbol | TGFBR2 |
| Protein Name | TGF-beta receptor type-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08917 (ecTbetaR2) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 144
- Clinical molecules 7
- Avg pChEMBL 6.66
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
- Transcriptional misregulation in cancer
Associated Diseases (6)
Active Molecules (144)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JZUKYILZIUEOPZ
|
6.7 | IC50 | 2 | — | |
LOWQGPGWACGUBU
|
6.7 | IC50 | 2 | — | |
MBGUKRYARWDEQD
|
6.7 | IC50 | 2 | — | |
OKWIIOORSZALCS
|
6.7 | IC50 | 2 | — | |
HNHLCXLNNWFVNS
|
6.6 | IC50 | 2 | — | |
RWIZWKXJKLBCDI
|
6.6 | IC50 | 2 | — | |
FAOGJKJCGFIFLI
|
6.6 | IC50 | 6 | — | |
OPGBVTXYOCNCFU
|
6.6 | IC50 | 2 | — | |
OSXBIOFAAZPBTB
|
6.6 | IC50 | 2 | — | |
USBMOTXWBABNGC
|
6.6 | IC50 | 2 | — | |
JGJFSDNRKJRVQG
|
6.6 | IC50 | 2 | — | |
MFAQYJIYDMLAIM
|
6.6 | Kd | 130 | Yes | |
QQWUGDVOUVUTOY
|
6.6 | Kd | 231 | Yes | |
ODPGGGTTYSGTGO
|
6.6 | Kd | 153 | — | |
HUCVSCRKTNYQEU
|
6.6 | IC50 | 2 | — | |
VAARYSWULJUGST
|
6.6 | Kd | 119 | Yes | |
BGASSDNBKMOKEZ
|
6.5 | IC50 | 2 | — | |
RAYASLMMTCQZGM
|
6.5 | IC50 | 2 | — | |
SHPFDGWALWEPGS
|
6.5 | Kd | 35 | — | |
BBDGBGOVJPEFBT
|
6.5 | IC50 | 6 | — | |
LNKMOULIMCFXDG
|
6.5 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
6.5 | Kd | 220 | — | |
WIBYDWSNIHNEPL
|
6.5 | IC50 | 2 | — | |
LDSCHZSRQSLWQV
|
6.5 | IC50 | 2 | — | |
SYCWRTUPLPDKDX
|
6.5 | IC50 | 3 | — | |
QNWFGJUQXVQTCF
|
6.4 | IC50 | 2 | — | |
MGCYGWOVPKUJBC
|
6.4 | IC50 | 2 | — | |
OZMSMXIUMHBELF
|
6.4 | IC50 | 2 | — | |
ACKBFDXVYCQQDK
|
6.4 | IC50 | 2 | — | |
GAWGUDTUQRRPQK
|
6.4 | IC50 | 2 | — | |
IBCXZJCWDGCXQT
|
6.4 | IC50 | 4 | — | |
IOMYOMXAQCULTN
|
6.4 | IC50 | 2 | — | |
JFAHUOXKADNXHK
|
6.4 | IC50 | 2 | — | |
FOVQNHTXUOXIEW
|
6.4 | IC50 | 2 | — | |
ZOFFXTKILIXKFI
|
6.4 | IC50 | 2 | — | |
GUBWWEPNZCJLMM
|
6.4 | IC50 | 2 | — | |
FVJODNBTCUGTJZ
|
6.3 | IC50 | 2 | — | |
QIPBSDCNDXMUCZ
|
6.3 | IC50 | 2 | — | |
BKZCTAIDOAKCRI
|
6.3 | IC50 | 2 | — | |
CATARNNGBNYRJP
|
6.3 | IC50 | 2 | — | |
UBTPOMHEYRBEHT
|
6.3 | IC50 | 5 | — | |
AOFAVFCOKNYJAU
|
6.3 | IC50 | 2 | — | |
KLPUMJUIPJTFRP
|
6.3 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
6.3 | Kd | 289 | Yes | |
BMMZGWDGXPPDEW
|
6.3 | IC50 | 2 | — | |
IRDIFSAZOXFGSK
|
6.2 | IC50 | 2 | — | |
AGMGRCAUAZCHPG
|
6.2 | IC50 | 5 | — | |
HULQVTAEMIYULR
|
6.2 | IC50 | 2 | — | |
NHXWKPGFUOSQCJ
|
6.2 | IC50 | 2 | — | |
NWZOSSQOJBZGSI
|
6.2 | IC50 | 2 | — |