Target Details
| UniProt AC | P37173 |
|---|---|
| Gene Symbol | TGFBR2 |
| Protein Name | TGF-beta receptor type-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08917 (ecTbetaR2) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 144
- Clinical molecules 7
- Avg pChEMBL 6.66
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
- Transcriptional misregulation in cancer
Associated Diseases (6)
Active Molecules (144)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PJNMAIKMKRLUIV
|
9.0 | IC50 | 3 | — | |
WCDLCPLAAKUJNY
|
8.9 | IC50 | 8 | — | |
QMOBMSIEJTZRFX
|
8.8 | IC50 | 2 | — | |
YSLKGORPFYLDEK
|
8.8 | IC50 | 2 | — | |
RGHVGCXGMWBBJX
|
8.4 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
8.2 | Kd | 1075 | — | |
GYHQCQQLLQAFGA
|
8.2 | IC50 | 2 | — | |
MTOKESMTTXYGSQ
|
8.2 | IC50 | 2 | — | |
WDNAXOPVZIEECR
|
7.8 | IC50 | 11 | — | |
GBOJIFPLPDQYNY
|
7.8 | IC50 | 2 | — | |
XBGWAKUQSRNWMA
|
7.8 | IC50 | 4 | — | |
GDGJWSLJIGCBGE
|
7.8 | IC50 | 2 | — | |
IIYOBXCNRFSCBH
|
7.8 | IC50 | 8 | — | |
SZVLDZCYMADNPG
|
7.6 | IC50 | 3 | — | |
ZBPTYYFUGHUNMQ
|
7.6 | IC50 | 2 | — | |
FBQRDQOHCIWKGC
|
7.4 | IC50 | 2 | — | |
WMTXIPYJYDISKM
|
7.4 | IC50 | 8 | — | |
XJYMAUIVMGKPRX
|
7.4 | IC50 | 2 | — | |
TZLMLVYIGMUVRJ
|
7.4 | IC50 | 2 | — | |
XODSKPZUYKGNMW
|
7.4 | IC50 | 2 | — | |
TXRZDWUIAYQQJI
|
7.3 | IC50 | 2 | — | |
OXAZKHAKYFXQPB
|
7.3 | IC50 | 2 | — | |
RAXZSEGXMBWYQK
|
7.3 | Kd | 21 | — | |
FHYUGAJXYORMHI
|
7.2 | IC50 | 7 | — | |
HJTMXUSRFLGCTK
|
7.2 | IC50 | 2 | — | |
FBMKNHDZOVPEAJ
|
7.2 | IC50 | 2 | — | |
DXVXGQDTEZKMLS
|
7.1 | IC50 | 2 | — | |
XLSYZSRXVVCHLS
|
7.1 | Kd | 48 | — | |
RXAXXPSLZPTWET
|
7.1 | IC50 | 2 | — | |
BQEUWLSQIXDQRX
|
7.0 | IC50 | 2 | — | |
WELLLPRMKHYPPA
|
7.0 | IC50 | 2 | — | |
XHBVYDAKJHETMP
|
7.0 | IC50 | 24 | Yes | |
BGASSDNBKMOKEZ
|
7.0 | IC50 | 2 | — | |
IRIRGFCFAMOTLN
|
6.9 | IC50 | 2 | — | |
ZPWIFPUPFCEENX
|
6.9 | IC50 | 2 | — | |
PZHBPITXMTZNSP
|
6.9 | IC50 | 2 | — | |
KBLQETSGJBJTIR
|
6.8 | IC50 | 2 | — | |
BYNUJHIHRYVHIS
|
6.8 | IC50 | 2 | — | |
YFNWWNRZJGMDBR
|
6.8 | Kd | 35 | — | |
CDOVNWNANFFLFJ
|
6.8 | IC50 | 10 | — | |
OFFLEANUVDDEBL
|
6.8 | IC50 | 2 | — | |
XTCPFWHYKZIXMD
|
6.8 | IC50 | 2 | — | |
CHAIHARSRAHKQQ
|
6.8 | IC50 | 2 | — | |
DBWYDBLIBRDZNH
|
6.8 | IC50 | 2 | — | |
RUBWYYYEDDAWLB
|
6.8 | IC50 | 5 | — | |
CSFVJUFNDCQAQO
|
6.7 | IC50 | 2 | — | |
IHLVSLOZUHKNMQ
|
6.7 | IC50 | 2 | — | |
JQZQDEAJANBRTM
|
6.7 | IC50 | 2 | — | |
OPHBHEKMLVUZBO
|
6.7 | IC50 | 2 | — | |
IOCHRHMTSUGIPK
|
6.7 | IC50 | 2 | — |