Target Details
| UniProt AC | P37023 |
|---|---|
| Gene Symbol | ACVRL1 |
| Protein Name | Activin receptor type-1-like |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 247
- Clinical molecules 7
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (247)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YCFHQBMHEXTGMF
|
6.6 | IC50 | 2 | — | |
GGQCWUKLPMFTDA
|
6.6 | IC50 | 5 | — | |
QPRFLHHDQOLCJS
|
6.6 | IC50 | 2 | — | |
BCCXLOMXYXXNIU
|
6.6 | IC50 | 2 | — | |
BAGWVDYVFGYURF
|
6.5 | IC50 | 2 | — | |
OVNAOUBDNBHVCI
|
6.5 | IC50 | 5 | — | |
RQXROVVCXFAAOM
|
6.5 | IC50 | 3 | — | |
DONRBWYKHKBNAQ
|
6.5 | IC50 | 2 | — | |
WBRIXUZLHYMBMA
|
6.5 | IC50 | 2 | — | |
NSVCYZBCJCPLDO
|
6.5 | IC50 | 2 | — | |
IOEZZOIIFUBFFP
|
6.5 | IC50 | 2 | — | |
RUBWYYYEDDAWLB
|
6.5 | IC50 | 5 | — | |
NNGJBTGAVCLGTM
|
6.5 | IC50 | 2 | — | |
GVKXHJBRWOYLAK
|
6.5 | IC50 | 3 | — | |
KPRPFTOLWQQUAV
|
6.5 | IC50 | 3 | — | |
STQMBDHGSGMKRK
|
6.5 | IC50 | 2 | — | |
ULQWBLKUEAKIFZ
|
6.5 | IC50 | 2 | — | |
FYPPBYUPMODRPA
|
6.5 | IC50 | 4 | — | |
LCNMZQCSKWYNQF
|
6.5 | IC50 | 2 | — | |
CLSVHDFWSGQNQH
|
6.5 | IC50 | 2 | — | |
HZMKNGJNPOBODV
|
6.4 | IC50 | 4 | — | |
OIDBPSOIVPMQGT
|
6.4 | IC50 | 2 | — | |
GAIBPGQSYNAFNN
|
6.4 | IC50 | 3 | — | |
PBPRYPLWJIJEMD
|
6.4 | IC50 | 2 | — | |
FVCQZDADSCVUOD
|
6.4 | IC50 | 2 | — | |
QNXUBBYNLLCNPH
|
6.4 | IC50 | 2 | — | |
GAIBPGQSYNAFNN
|
6.4 | IC50 | 3 | — | |
JUACWTBEXKUOOV
|
6.4 | IC50 | 2 | — | |
LJUBHCPBQBKBHM
|
6.4 | IC50 | 5 | — | |
HIWHLPKRUZGHRR
|
6.4 | IC50 | 4 | — | |
JWSRLZGLCYGKSQ
|
6.4 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
6.3 | Kd | 102 | Yes | |
UHTHHESEBZOYNR
|
6.3 | Kd | 66 | Yes | |
UVOJVOHBYLNVCM
|
6.3 | IC50 | 2 | — | |
KIUMBIWMXBUHDW
|
6.3 | IC50 | 3 | — | |
CCKKGJFQFLRASM
|
6.3 | IC50 | 2 | — | |
FZJGVHATMCAPLO
|
6.3 | IC50 | 5 | — | |
HZFKGEGMOFIQKL
|
6.3 | IC50 | 2 | — | |
BXMKDTWGFLBPKB
|
6.3 | IC50 | 2 | — | |
PBPRYPLWJIJEMD
|
6.3 | IC50 | 2 | — | |
AJIRLUWVMCLWFU
|
6.3 | IC50 | 2 | — | |
FTSHNQVAJPKPPY
|
6.3 | IC50 | 2 | — | |
MDGXLOFLFFEXSH
|
6.3 | IC50 | 2 | — | |
VUEWHTWKZUEQMF
|
6.3 | IC50 | 4 | — | |
KPRPFTOLWQQUAV
|
6.3 | IC50 | 2 | — | |
NTLWKKILBCETHV
|
6.3 | IC50 | 4 | — | |
SQRAKIQIMGAALF
|
6.3 | IC50 | 2 | — | |
DBAUTMSTTOYZCH
|
6.3 | IC50 | 2 | — | |
QKGNJQNQCKFAFD
|
6.3 | IC50 | 2 | — | |
SRPLSQLPBCVKSL
|
6.2 | IC50 | 2 | — |