Target Details
| UniProt AC | P37023 |
|---|---|
| Gene Symbol | ACVRL1 |
| Protein Name | Activin receptor type-1-like |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 247
- Clinical molecules 7
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (247)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BZXHYPDAQAEAKY
|
7.4 | IC50 | 5 | — | |
CNEUJSQUCXSRDD
|
7.4 | Kd | 7 | — | |
LYZXDNCSIHIAMI
|
7.4 | IC50 | 3 | — | |
JDYMCSKANXEKMK
|
7.4 | IC50 | 3 | — | |
WCDLCPLAAKUJNY
|
7.4 | IC50 | 8 | — | |
XQLHGVZYEZLJEG
|
7.4 | IC50 | 3 | — | |
PRKWSDOLROTYLX
|
7.3 | IC50 | 3 | — | |
SRIVDECCESIDAQ
|
7.3 | IC50 | 3 | — | |
FVRYPYDPKSZGNS
|
7.3 | IC50 | 2 | — | |
WOKJIIMDDCFJJH
|
7.3 | IC50 | 2 | — | |
GLJHPFGWEFTXKS
|
7.3 | IC50 | 2 | — | |
RZYYJEYQNNJBMD
|
7.3 | IC50 | 3 | — | |
IBCXZJCWDGCXQT
|
7.3 | IC50 | 4 | — | |
IPESYYFOXATSFJ
|
7.3 | IC50 | 3 | — | |
IIYOBXCNRFSCBH
|
7.3 | IC50 | 8 | — | |
UXVFRKCJRULCNV
|
7.3 | IC50 | 4 | — | |
ODVUZZFWFOPOAH
|
7.3 | IC50 | 5 | — | |
WMTXIPYJYDISKM
|
7.3 | IC50 | 8 | — | |
QQWUGDVOUVUTOY
|
7.2 | Kd | 231 | Yes | |
MNCBGNHYCLQCSA
|
7.2 | IC50 | 2 | — | |
QPIFMCLNACVAAT
|
7.2 | IC50 | 7 | — | |
VAARYSWULJUGST
|
7.2 | Kd | 119 | Yes | |
QCEHAYINFMPPPM
|
7.1 | IC50 | 3 | — | |
PVDWNOWJXDXMDH
|
7.1 | IC50 | 5 | — | |
ZCFRPQTXMMLPFH
|
7.1 | IC50 | 2 | — | |
FCURQEMLQWEPFI
|
7.1 | IC50 | 2 | — | |
OVXMCCQKIOSDGE
|
7.1 | IC50 | 3 | — | |
ABEPADPRAQLNSN
|
7.1 | IC50 | 3 | — | |
DPDIGSURNQRYQS
|
7.1 | IC50 | 3 | — | |
JFDSOYMKCLUKEJ
|
7.0 | IC50 | 2 | — | |
LMNXBEZQGBWMMY
|
7.0 | IC50 | 3 | — | |
UBTPOMHEYRBEHT
|
7.0 | IC50 | 5 | — | |
UTCHZVUDAGSGMY
|
7.0 | IC50 | 3 | — | |
HZFKGEGMOFIQKL
|
7.0 | IC50 | 2 | — | |
IEJPGJXAWUJROQ
|
7.0 | IC50 | 5 | — | |
YTUZELSDHUVEFM
|
7.0 | IC50 | 4 | — | |
BBWFHMVFMVFXJP
|
7.0 | IC50 | 3 | — | |
JHBVJUXBKKKJGW
|
7.0 | IC50 | 2 | — | |
UAHBMBZHEHEEAW
|
7.0 | IC50 | 4 | — | |
XHBVYDAKJHETMP
|
7.0 | IC50 | 24 | Yes | |
DONRBWYKHKBNAQ
|
7.0 | IC50 | 2 | — | |
QDSMDFVMOMUBDR
|
7.0 | IC50 | 2 | — | |
JXPPULPLYFLFJI
|
6.9 | IC50 | 3 | — | |
MOTRKLJWPDOTBN
|
6.9 | IC50 | 3 | — | |
RIGIHWPKCOSNDD
|
6.9 | IC50 | 3 | — | |
QIXWNWRGNUGMRT
|
6.9 | IC50 | 2 | — | |
QXPNJMHRUZCEAP
|
6.9 | IC50 | 14 | — | |
NJSRQYMTTJJEJH
|
6.9 | IC50 | 2 | — | |
WCTODNJGIAJWJX
|
6.9 | IC50 | 2 | — | |
GPLMXGSESNBQQL
|
6.9 | IC50 | 2 | — |