Target Details
| UniProt AC | P37023 |
|---|---|
| Gene Symbol | ACVRL1 |
| Protein Name | Activin receptor type-1-like |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 247
- Clinical molecules 7
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (247)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.9 | IC50 | 118 | — | |
CJLMANFTWLNAKC
|
8.7 | IC50 | 5 | — | |
MFAQYJIYDMLAIM
|
8.5 | Kd | 130 | Yes | |
MQFUFNHTCJRLKW
|
8.4 | IC50 | 6 | — | |
WJASKODGMHBDFO
|
8.4 | IC50 | 5 | — | |
LRJJEMRURFIKDD
|
8.3 | IC50 | 6 | — | |
SHWKNOUREYUNBF
|
8.2 | IC50 | 6 | — | |
KIAKJNRDKPGTQR
|
8.2 | IC50 | 6 | — | |
BNPMMVDYMYENIM
|
8.0 | IC50 | 4 | — | |
FOLXFWBVNHRGIV
|
8.0 | IC50 | 6 | — | |
SCHRCCHASZMVAB
|
8.0 | IC50 | 7 | — | |
WOAXRKYXUKTLEM
|
8.0 | IC50 | 7 | — | |
QQYOZULVMVWDFQ
|
8.0 | IC50 | 3 | — | |
WTMROIBZVGJXRP
|
8.0 | IC50 | 4 | — | |
FFLJVBPCONQSQW
|
7.9 | IC50 | 8 | — | |
CDOVNWNANFFLFJ
|
7.9 | IC50 | 10 | — | |
DPMQHTABGLRCQK
|
7.8 | IC50 | 5 | — | |
BBDGBGOVJPEFBT
|
7.8 | IC50 | 6 | — | |
ZUSOUYHYDDCGIC
|
7.8 | IC50 | 4 | — | |
DUGKWSLUPDXHDO
|
7.8 | IC50 | 3 | — | |
LKQSELSKVLDVHG
|
7.8 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
7.8 | Kd | 97 | Yes | |
RKBYYWVZFBATHQ
|
7.8 | IC50 | 12 | — | |
UDXFCKQHYWOCHB
|
7.8 | IC50 | 2 | — | |
RIWTUJFFSTVYPW
|
7.8 | IC50 | 6 | — | |
UPBPVAZUFAXUAC
|
7.8 | IC50 | 6 | — | |
FHTCHCUICJOIGJ
|
7.8 | IC50 | 7 | — | |
AJRCHNXNYNADRQ
|
7.8 | IC50 | 3 | — | |
GIAGHNVPQYZDIK
|
7.8 | IC50 | 3 | — | |
MXDCACLUETVZNL
|
7.7 | IC50 | 8 | — | |
PAHLIVNOHVHPBG
|
7.7 | IC50 | 6 | — | |
CXZJXVJPISUKMR
|
7.7 | IC50 | 6 | — | |
XYIZJZFZXCURDK
|
7.7 | IC50 | 5 | — | |
JDAFKLSYNCTYHC
|
7.6 | IC50 | 3 | — | |
XBJCMGUGQRINQY
|
7.6 | IC50 | 2 | — | |
HSAUZUYGDAHMLS
|
7.6 | IC50 | 2 | — | |
XJRNYUDHNXZYCF
|
7.6 | IC50 | 3 | — | |
ZOMQASFZVQEKHR
|
7.6 | IC50 | 3 | — | |
FAOGJKJCGFIFLI
|
7.6 | IC50 | 6 | — | |
BHUXVRVMMYAXKN
|
7.6 | IC50 | 3 | — | |
JMIFGARJSWXZSH
|
7.6 | IC50 | 3 | — | |
QCXBJMRMYRQRCV
|
7.6 | IC50 | 4 | — | |
WSNLCMQIUFLQBS
|
7.6 | IC50 | 3 | — | |
NTZZVPFINNIFIF
|
7.5 | IC50 | 2 | — | |
ZBOSAPQCJDMZCV
|
7.5 | IC50 | 6 | — | |
WJSYQJFCHPTVCI
|
7.5 | IC50 | 3 | — | |
KVLSZJPFQDRDPI
|
7.4 | IC50 | 4 | — | |
KVDFCDPSKGACEZ
|
7.4 | IC50 | 4 | — | |
NQAMVBJCWLPNJI
|
7.4 | IC50 | 2 | — | |
OBLCGNSTBZOGIQ
|
7.4 | IC50 | 3 | — |