Target Details
| UniProt AC | P36897 |
|---|---|
| Gene Symbol | TGFBR1 |
| Protein Name | TGF-beta receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 428
- Clinical molecules 14
- Avg pChEMBL 7.75
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Apelin signaling pathway
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
Associated Diseases (3)
Active Molecules (428)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GGQCWUKLPMFTDA
|
6.2 | IC50 | 5 | — | |
LJUBHCPBQBKBHM
|
6.2 | IC50 | 5 | — | |
GFEAXKZXFORDDU
|
6.2 | IC50 | 2 | — | |
BZXHYPDAQAEAKY
|
6.2 | IC50 | 5 | — | |
SOAGPOPZDBBHMB
|
6.2 | IC50 | 2 | — | |
FZJGVHATMCAPLO
|
6.2 | IC50 | 5 | — | |
HRKJFKJZUNJKNU
|
6.2 | IC50 | 10 | — | |
OVNAOUBDNBHVCI
|
6.2 | IC50 | 5 | — | |
PJNMAIKMKRLUIV
|
6.2 | IC50 | 3 | — | |
YPTIRJISDXITNF
|
6.2 | IC50 | 3 | — | |
GVISBDZSDFJHJS
|
6.1 | IC50 | 3 | — | |
ROCFHKYAFOQDHC
|
6.1 | IC50 | 5 | — | |
UBTPOMHEYRBEHT
|
6.1 | IC50 | 5 | — | |
IRAQZZSMFOUNQT
|
6.1 | IC50 | 2 | — | |
JROFGZPOBKIAEW
|
6.1 | Kd | 10 | — | |
OFCHEKHQCUGWFP
|
6.1 | IC50 | 2 | — | |
HDMLUZMVBVBTJX
|
6.1 | IC50 | 2 | — | |
ZRCZZPPDWCVIOL
|
6.1 | IC50 | 2 | — | |
JFQHZKYTJUOQDK
|
6.1 | IC50 | 2 | — | |
NYYYLFUSXWJOML
|
6.1 | IC50 | 3 | — | |
ODVUZZFWFOPOAH
|
6.0 | IC50 | 5 | — | |
CNEUJSQUCXSRDD
|
6.0 | Kd | 7 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KTEIFNKAUNYNJU
|
6.0 | Kd | 114 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MZIQJPGLZXVJCP
|
6.0 | IC50 | 2 | — | |
VUEWHTWKZUEQMF
|
6.0 | IC50 | 4 | — |