Target Details
| UniProt AC | P36897 |
|---|---|
| Gene Symbol | TGFBR1 |
| Protein Name | TGF-beta receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 428
- Clinical molecules 14
- Avg pChEMBL 7.75
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Apelin signaling pathway
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
Associated Diseases (3)
Active Molecules (428)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XMGRGPZCVNKAOK
|
7.3 | IC50 | 2 | — | |
OXAUEWLYSXHBDP
|
7.2 | IC50 | 2 | — | |
CPYLRRTWXCUAOG
|
7.2 | IC50 | 2 | — | |
MQFUFNHTCJRLKW
|
7.2 | IC50 | 6 | — | |
CCODMHGTAFMNHJ
|
7.2 | IC50 | 2 | — | |
CKLULXBYHFYPHR
|
7.2 | IC50 | 2 | — | |
CRLKMDIFJAUNGQ
|
7.2 | IC50 | 2 | — | |
KHPXUXMWUXXXLH
|
7.2 | IC50 | 2 | — | |
VLWLLXSQJNQRJG
|
7.2 | IC50 | 2 | — | |
AQPVZDUZQVWOEP
|
7.2 | IC50 | 3 | — | |
LZKXCQQNNYURRI
|
7.2 | IC50 | 2 | — | |
JCBZLQOFQWJOBF
|
7.2 | IC50 | 2 | — | |
WGALZWWKJHCIBC
|
7.2 | IC50 | 3 | — | |
CGAOZJWPBAWCGJ
|
7.1 | IC50 | 2 | — | |
XBGWAKUQSRNWMA
|
7.1 | IC50 | 4 | — | |
CQFMEEGANZACLR
|
7.1 | IC50 | 3 | — | |
FHRZBVSUXBSDPP
|
7.1 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
7.1 | Kd | 97 | Yes | |
YWKTUNHCMPHUCG
|
7.1 | IC50 | 3 | — | |
FDMRIXRWLAMVEF
|
7.1 | IC50 | 2 | — | |
NLJVTJDPRBIFFV
|
7.1 | IC50 | 3 | — | |
SYCWRTUPLPDKDX
|
7.1 | IC50 | 3 | — | |
AMZUNRUJZDTWPE
|
7.1 | IC50 | 2 | — | |
DLXGDQAWZVGPQU
|
7.1 | IC50 | 2 | — | |
KXUIBHJQCVWSNW
|
7.1 | IC50 | 2 | — | |
RRSMQTBPLPCBAN
|
7.1 | IC50 | 3 | — | |
SGMXHEIWJQTVMJ
|
7.1 | IC50 | 3 | — | |
FHYUGAJXYORMHI
|
7.0 | IC50 | 7 | — | |
SCHRCCHASZMVAB
|
7.0 | IC50 | 7 | — | |
DDVZCQMFWBEKAW
|
7.0 | IC50 | 2 | — | |
DSJFEZATROEIML
|
7.0 | IC50 | 2 | — | |
MFAQYJIYDMLAIM
|
7.0 | Kd | 130 | Yes | |
MXDCACLUETVZNL
|
7.0 | IC50 | 8 | — | |
AOTADNCHLKUEAX
|
7.0 | IC50 | 2 | — | |
CXFUMQXKEITWKR
|
7.0 | IC50 | 2 | — | |
IVRXNBXKWIJUQB
|
6.9 | IC50 | 10 | — | |
UIARLYUEJFELEN
|
6.9 | Kd | 289 | Yes | |
XCQPASNBVLQPAI
|
6.9 | IC50 | 2 | — | |
IRFYJXPFDRTUSQ
|
6.9 | IC50 | 2 | — | |
LRSOQWKCWLRMRR
|
6.9 | IC50 | 2 | — | |
SJOCBUINMBQCTH
|
6.9 | IC50 | 2 | — | |
XIAQAOWQYMNJJB
|
6.9 | IC50 | 2 | — | |
DKZYXHCYPUVGAF
|
6.8 | Kd | 112 | — | |
DERIBTSHHPNLEG
|
6.8 | IC50 | 2 | — | |
FFEWOBPMLFVMPC
|
6.8 | IC50 | 2 | — | |
IKJMJDPMGHFSNH
|
6.8 | IC50 | 2 | — | |
OTMZESJOOWWVGH
|
6.8 | IC50 | 2 | — | |
LKZOWZZOQPWIFO
|
6.8 | IC50 | 2 | — | |
SZVLDZCYMADNPG
|
6.8 | IC50 | 3 | — | |
DPDGLGMFKKTTPN
|
6.7 | IC50 | 2 | — |