Target Details
| UniProt AC | P36897 |
|---|---|
| Gene Symbol | TGFBR1 |
| Protein Name | TGF-beta receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 428
- Clinical molecules 14
- Avg pChEMBL 7.75
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Apelin signaling pathway
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
Associated Diseases (3)
Active Molecules (428)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NVZWXPUBNZUNFM
|
7.6 | IC50 | 2 | — | |
PVBJXPIQVPYBQR
|
7.6 | IC50 | 2 | — | |
GVDHTILDVBEBLW
|
7.5 | IC50 | 2 | — | |
NRNOAZUAWDMPFI
|
7.5 | IC50 | 2 | — | |
QRINOTMCPQYUCC
|
7.5 | IC50 | 2 | — | |
QRINOTMCPQYUCC
|
7.5 | IC50 | 2 | — | |
COKRWYWHAZQZLD
|
7.5 | IC50 | 2 | — | |
CTCRBAORDBWNPN
|
7.5 | IC50 | 2 | — | |
DOBRZXIRNFXQCN
|
7.5 | IC50 | 2 | — | |
NLIQPLLQHGVUIO
|
7.5 | IC50 | 2 | — | |
MJWOMIHVCXLYLG
|
7.5 | IC50 | 2 | — | |
PRPWREAEINLLOR
|
7.5 | IC50 | 2 | — | |
BVWNOAMYVMKTGC
|
7.5 | IC50 | 3 | — | |
YOLJORSLLBNCFO
|
7.5 | IC50 | 2 | — | |
ILRGLUAABODDJU
|
7.5 | IC50 | 3 | — | |
AOWURAHNMNLYFX
|
7.5 | IC50 | 2 | — | |
KLPUMJUIPJTFRP
|
7.5 | IC50 | 2 | — | |
MJWGUTNEFRSROZ
|
7.5 | IC50 | 2 | — | |
CJTQBCMGMLTHPI
|
7.5 | IC50 | 4 | — | |
JEMYLFFKZOOMQU
|
7.5 | IC50 | 2 | — | |
MUSRTIADFPCYTQ
|
7.5 | IC50 | 2 | — | |
NXDCVJJDDFFEON
|
7.5 | IC50 | 2 | — | |
OGPVQKHTKOAKDQ
|
7.5 | IC50 | 2 | — | |
ATSRJSICZUBQJU
|
7.5 | IC50 | 2 | — | |
GUDFYAAWBWHCJA
|
7.5 | IC50 | 2 | — | |
JVOASSRFSRQUDN
|
7.5 | IC50 | 2 | — | |
MHWCSGRDASEMOM
|
7.5 | IC50 | 2 | — | |
AIQDEVOVNXQXKX
|
7.5 | IC50 | 2 | — | |
QRINOTMCPQYUCC
|
7.4 | IC50 | 2 | — | |
MOXKDKRBVAMLRS
|
7.4 | IC50 | 3 | — | |
QLCHJBPDLYRMBA
|
7.4 | IC50 | 2 | — | |
GGVVKPVKOVIANA
|
7.4 | IC50 | 2 | — | |
SRVVCPDKVNJPAH
|
7.4 | IC50 | 2 | — | |
VVEMGKLSOKWLEB
|
7.4 | IC50 | 2 | — | |
LUJQZBILMIUCPF
|
7.3 | IC50 | 2 | — | |
DJWQPNVQFDNUSO
|
7.3 | IC50 | 2 | — | |
LBZFXCHCPXGOBO
|
7.3 | IC50 | 2 | — | |
QNZSQJBDZIOEAN
|
7.3 | IC50 | 2 | — | |
BERLXWPRSBJFHO
|
7.3 | IC50 | 4 | — | |
NPKLXIBDXVXQBM
|
7.3 | IC50 | 2 | — | |
YESUBTROVJOXSV
|
7.3 | IC50 | 3 | — | |
IBCXZJCWDGCXQT
|
7.3 | IC50 | 4 | — | |
IHLVSLOZUHKNMQ
|
7.3 | IC50 | 2 | — | |
QGMSQMSDEUEWCM
|
7.3 | IC50 | 2 | — | |
IRNKSUFVVQZURD
|
7.3 | IC50 | 2 | — | |
WOAXRKYXUKTLEM
|
7.3 | IC50 | 7 | — | |
FIGRKDLMTBPIFC
|
7.3 | IC50 | 2 | — | |
TWYFELLCKHAKCY
|
7.3 | IC50 | 2 | — | |
WGZOTBUYUFBEPZ
|
7.3 | IC50 | 4 | — | |
XMGRGPZCVNKAOK
|
7.3 | IC50 | 2 | — |