Target Details
| UniProt AC | P36897 |
|---|---|
| Gene Symbol | TGFBR1 |
| Protein Name | TGF-beta receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 428
- Clinical molecules 14
- Avg pChEMBL 7.75
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Apelin signaling pathway
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
Associated Diseases (3)
Active Molecules (428)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZOFFXTKILIXKFI
|
7.8 | IC50 | 2 | — | |
IVGZZSIANNYXTI
|
7.8 | IC50 | 2 | — | |
OCJCDFHRNVHPGQ
|
7.8 | IC50 | 2 | — | |
ODWRQIDMGOOEIE
|
7.8 | IC50 | 2 | — | |
POPIUCWMQJYOGO
|
7.8 | IC50 | 2 | — | |
ZMUWOLHXXFLWAH
|
7.8 | IC50 | 2 | — | |
DTWRYSLEWSOAST
|
7.8 | IC50 | 2 | — | |
GIXYMNJSHSCLBB
|
7.8 | IC50 | 2 | — | |
OAYQAXXBPMOPLN
|
7.8 | IC50 | 2 | — | |
OXVQEZJDLGHTQA
|
7.8 | IC50 | 2 | — | |
UXFTVPGMWIESDP
|
7.8 | IC50 | 2 | — | |
ZPWWHJQTSTXJOQ
|
7.8 | IC50 | 2 | — | |
HPZDDBNHJHAGNV
|
7.8 | IC50 | 2 | — | |
RYKSGWSKILPDDY
|
7.8 | IC50 | 4 | — | |
CKODUGCWZCWIRZ
|
7.8 | IC50 | 2 | — | |
NRALVILIKBNNQX
|
7.8 | IC50 | 2 | — | |
SAGZIBJAQGBRQA
|
7.8 | IC50 | 2 | — | |
FKBBYKXWULFABH
|
7.7 | IC50 | 2 | — | |
HUCVSCRKTNYQEU
|
7.7 | IC50 | 2 | — | |
LOWQGPGWACGUBU
|
7.7 | IC50 | 2 | — | |
YLJGNMFEAJARMT
|
7.7 | IC50 | 2 | — | |
KXQAYIADFSNSAJ
|
7.7 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.7 | Kd | 1075 | — | |
JZVPITOQWJPGIA
|
7.7 | IC50 | 2 | — | |
MMWRLDUOCZWADE
|
7.7 | IC50 | 2 | — | |
NKEPPANSOKDJCW
|
7.7 | IC50 | 3 | — | |
ZMDZLOKVZATBIJ
|
7.7 | IC50 | 2 | — | |
REHNTCRUPYALSU
|
7.7 | IC50 | 2 | — | |
IXHWEVQIYXKCCA
|
7.7 | IC50 | 2 | — | |
JLZZQIDAVCRRTQ
|
7.7 | IC50 | 2 | — | |
MTOKESMTTXYGSQ
|
7.7 | IC50 | 2 | — | |
VMAJWCRBVRIZQR
|
7.7 | IC50 | 2 | — | |
UARGTFDABIYTIP
|
7.6 | IC50 | 3 | — | |
LLPMPHUIFSJZAT
|
7.6 | IC50 | 2 | — | |
LMAUBLPXDXVPSK
|
7.6 | IC50 | 2 | — | |
UVBZZXVKQPKWOZ
|
7.6 | IC50 | 2 | — | |
XJYMAUIVMGKPRX
|
7.6 | IC50 | 2 | — | |
ZJRZWWGSQJZWFS
|
7.6 | IC50 | 2 | — | |
IJHZZNGTHXCEFT
|
7.6 | IC50 | 2 | — | |
IOMYOMXAQCULTN
|
7.6 | IC50 | 2 | — | |
IPBLCOKXDQHSQW
|
7.6 | IC50 | 2 | — | |
NWKVJLWADKJMIM
|
7.6 | IC50 | 2 | — | |
JIJYWPGTRDMEFZ
|
7.6 | IC50 | 5 | Yes | |
KJTYZDORHCDZPS
|
7.6 | IC50 | 2 | — | |
LVEUPFUJRKZPEN
|
7.6 | IC50 | 2 | — | |
SXNCFFITOIFUMU
|
7.6 | IC50 | 2 | — | |
XNECSXXXAVERCS
|
7.6 | IC50 | 2 | — | |
YVNIRHOSELPYAW
|
7.6 | IC50 | 2 | — | |
UNKRRNQGTJWRNM
|
7.6 | IC50 | 2 | — | |
KIAKJNRDKPGTQR
|
7.6 | IC50 | 6 | — |