Target Details
| UniProt AC | P36897 |
|---|---|
| Gene Symbol | TGFBR1 |
| Protein Name | TGF-beta receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 428
- Clinical molecules 14
- Avg pChEMBL 7.75
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Apelin signaling pathway
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
Associated Diseases (3)
Active Molecules (428)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PNNHSDGMXFKVRN
|
8.1 | IC50 | 2 | — | |
ZIFZTQMNCSFVKL
|
8.1 | IC50 | 2 | — | |
BIRMNZNMTFDQFC
|
8.1 | IC50 | 2 | — | |
BPRNIBFKCRFPOU
|
8.1 | IC50 | 2 | — | |
CKNHHTRTDCIBGT
|
8.1 | IC50 | 2 | — | |
CQITVCPBOHXPEG
|
8.1 | IC50 | 2 | — | |
CSMOUVFWIWCQLV
|
8.1 | IC50 | 2 | — | |
JZOMCUFMJKGTSX
|
8.1 | IC50 | 2 | — | |
VBECRVQGKLDJIE
|
8.1 | IC50 | 2 | — | |
YXUCEYHUMMDUOT
|
8.1 | IC50 | 2 | — | |
AAXTYXQSGJCLLL
|
8.0 | IC50 | 2 | — | |
COZUKVUBSCQZGM
|
8.0 | IC50 | 2 | — | |
CBDNDJPIMQLOAF
|
8.0 | IC50 | 2 | — | |
HZKLJOMOWASAJL
|
8.0 | IC50 | 2 | — | |
RRDBKKJRGDARIV
|
8.0 | IC50 | 2 | — | |
ICADYKQQHFVDME
|
8.0 | Kd | 2 | — | |
KJUCPVIVNLPLEE
|
8.0 | IC50 | 10 | — | |
LEYBPKZGESRTRA
|
8.0 | IC50 | 2 | — | |
NYCBVTAWFSXLGH
|
8.0 | IC50 | 2 | — | |
RNKGUQCZUZXJAW
|
8.0 | IC50 | 2 | — | |
WETVZDDFVHQTTQ
|
8.0 | IC50 | 2 | — | |
JQZGDZPOTURSKE
|
8.0 | IC50 | 2 | — | |
PZHBPITXMTZNSP
|
8.0 | IC50 | 2 | — | |
WQPRHDZTTYJDPW
|
8.0 | IC50 | 2 | — | |
BWCGKHAXQRCBGT
|
8.0 | IC50 | 2 | — | |
QPFVXQGTWSDAJK
|
8.0 | IC50 | 3 | — | |
RPJBEJCOQGUCJS
|
8.0 | IC50 | 2 | — | |
DSKSACIENVKOMV
|
8.0 | IC50 | 2 | — | |
GSCVYTUEFYPEHY
|
8.0 | IC50 | 2 | — | |
ZJHPTJJPYYJHCT
|
7.9 | IC50 | 2 | — | |
BTEPRNNLWBMDPC
|
7.9 | IC50 | 2 | — | |
GHMASSBRZQUWTC
|
7.9 | IC50 | 2 | — | |
HIFGZZBMONHQCC
|
7.9 | IC50 | 2 | — | |
SVFWZNDJPVECNU
|
7.9 | IC50 | 2 | — | |
FJCDSQATIJKQKA
|
7.9 | IC50 | 5 | — | |
GUBWWEPNZCJLMM
|
7.9 | IC50 | 2 | — | |
ISSKIYXWEWUJFS
|
7.9 | IC50 | 2 | — | |
OWIYYKSTVQMPLM
|
7.9 | IC50 | 2 | — | |
TVJUAWATEKXUSU
|
7.9 | IC50 | 2 | — | |
RWKUOBJGDXCOKM
|
7.9 | IC50 | 2 | — | |
CGEGHLLVXRIRQP
|
7.8 | IC50 | 2 | — | |
HHGCXYQSDOHURD
|
7.8 | IC50 | 2 | — | |
IQOTVGHBBHOBKR
|
7.8 | IC50 | 2 | — | |
VYTQMUCONGRNBX
|
7.8 | IC50 | 3 | — | |
YJKNBYBEJYUUHW
|
7.8 | IC50 | 2 | — | |
YTBQDRNYIQRKTK
|
7.8 | IC50 | 2 | — | |
NVUCXTBAGHPGKH
|
7.8 | IC50 | 2 | — | |
OXSDTRSIBXBIJL
|
7.8 | IC50 | 2 | — | |
POMBIFQUJUHXAV
|
7.8 | IC50 | 2 | — | |
XYCSMDDTSMSRGN
|
7.8 | IC50 | 2 | — |