Target Details
| UniProt AC | P36897 |
|---|---|
| Gene Symbol | TGFBR1 |
| Protein Name | TGF-beta receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 428
- Clinical molecules 14
- Avg pChEMBL 7.75
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Apelin signaling pathway
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
Associated Diseases (3)
Active Molecules (428)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XODSKPZUYKGNMW
|
8.5 | IC50 | 2 | — | |
ZYSFQPYDGIWDSA
|
8.5 | IC50 | 2 | — | |
XHCKXJQTGAAHKU
|
8.5 | IC50 | 2 | — | |
GZOYOEIHAGHGFM
|
8.5 | IC50 | 6 | — | |
QNWFGJUQXVQTCF
|
8.5 | IC50 | 2 | — | |
HUEXJRRSSHIGFJ
|
8.5 | IC50 | 2 | — | |
LHYODZLDZIQFCQ
|
8.5 | IC50 | 2 | — | |
CSFVJUFNDCQAQO
|
8.4 | IC50 | 2 | — | |
SZPOIQZUDFAZMU
|
8.4 | IC50 | 2 | — | |
QCEHAYINFMPPPM
|
8.4 | IC50 | 3 | — | |
JXKHBWPSMRRQQD
|
8.4 | IC50 | 2 | — | |
UARGTFDABIYTIP
|
8.4 | IC50 | 2 | — | |
WOKGXNSTAOLINW
|
8.4 | IC50 | 2 | — | |
YQSRHUJKRYNBHZ
|
8.4 | IC50 | 2 | — | |
WDNAXOPVZIEECR
|
8.4 | IC50 | 11 | — | |
DGTYEYRETGUTQA
|
8.4 | IC50 | 2 | — | |
NIQVUPWBHUGPKD
|
8.4 | IC50 | 2 | — | |
FFCNMKMMYJYENY
|
8.3 | IC50 | 2 | — | |
BKZCTAIDOAKCRI
|
8.3 | IC50 | 2 | — | |
RARPNWVPJDMGQD
|
8.3 | IC50 | 2 | — | |
DPPWGFZLKKSGLV
|
8.3 | IC50 | 2 | — | |
BVTHZDXMHJBZAJ
|
8.3 | IC50 | 2 | — | |
FIGWQDHDUNOAHY
|
8.3 | IC50 | 2 | — | |
FXRXNBVYNBHKIT
|
8.3 | IC50 | 2 | — | |
HXHAJRMTJXHJJZ
|
8.3 | Kd | 52 | Yes | |
IHPNHLBHEBHRGJ
|
8.3 | IC50 | 2 | — | |
RWBHBQMJZIBEBQ
|
8.3 | IC50 | 2 | — | |
YOKGFEAEVZNOAR
|
8.2 | IC50 | 5 | — | |
CEXJBZFYQTYDOL
|
8.2 | IC50 | 2 | — | |
JSICPTDRMBTMON
|
8.2 | IC50 | 2 | — | |
NLTJLIGESBNQSN
|
8.2 | IC50 | 2 | — | |
HESAPDRVFTXZTE
|
8.2 | IC50 | 2 | — | |
MFIQSIKORGZOQM
|
8.2 | IC50 | 2 | — | |
NUVPAWNZKYSCFY
|
8.2 | IC50 | 2 | — | |
WKDQUOATEFNKLP
|
8.2 | IC50 | 2 | — | |
BRFBWBYMLHDXOU
|
8.2 | IC50 | 2 | — | |
DJQVUYJBUCHJDH
|
8.2 | IC50 | 2 | — | |
OIYYETCFCIAZSC
|
8.2 | IC50 | 2 | — | |
PRGJXCHZTFKJNC
|
8.2 | IC50 | 2 | — | |
WKOVMPFJSORYMW
|
8.2 | IC50 | 2 | — | |
XETRNBBNUVDOJG
|
8.2 | IC50 | 2 | — | |
MCKOAFYHBBPGJY
|
8.1 | IC50 | 2 | — | |
VXRUZPWNIPZAQV
|
8.1 | IC50 | 2 | — | |
GFYMGKKOEOHJOB
|
8.1 | IC50 | 2 | — | |
GXSVCLUDQARGGX
|
8.1 | IC50 | 2 | — | |
PXKXNBMBKGONPB
|
8.1 | IC50 | 2 | — | |
ZUUYXUJYVRIKRA
|
8.1 | IC50 | 2 | — | |
FBMKNHDZOVPEAJ
|
8.1 | IC50 | 2 | — | |
JJYZCPRITYKJAQ
|
8.1 | IC50 | 2 | — | |
YGLGBLUEVWJWHB
|
8.1 | IC50 | 2 | — |