Target Details
| UniProt AC | P36897 |
|---|---|
| Gene Symbol | TGFBR1 |
| Protein Name | TGF-beta receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 428
- Clinical molecules 14
- Avg pChEMBL 7.75
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Apelin signaling pathway
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
Associated Diseases (3)
Active Molecules (428)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FGCSLJAOHVQQFY
|
9.0 | IC50 | 2 | — | |
HNHLCXLNNWFVNS
|
9.0 | IC50 | 2 | — | |
IMPLASSOUGGFTO
|
9.0 | IC50 | 2 | — | |
MPUBMJCSEANNKB
|
9.0 | IC50 | 2 | — | |
NZEXAUMJUOFREM
|
9.0 | IC50 | 2 | — | |
XGYKDWXVWCPZML
|
9.0 | IC50 | 2 | — | |
AOFAVFCOKNYJAU
|
9.0 | IC50 | 2 | — | |
STPUEPLVTCNYHC
|
9.0 | IC50 | 2 | — | |
TZLMLVYIGMUVRJ
|
9.0 | IC50 | 2 | — | |
HJZCMIKTRDMVQA
|
8.9 | IC50 | 2 | — | |
MGPDWDBEWFYGJF
|
8.9 | IC50 | 2 | — | |
QIPBSDCNDXMUCZ
|
8.9 | IC50 | 2 | — | |
SXDZOHOHBPOZQD
|
8.9 | IC50 | 2 | — | |
XTCPFWHYKZIXMD
|
8.9 | IC50 | 2 | — | |
CSFCQZGWCYRHAU
|
8.9 | IC50 | 2 | — | |
DEBKOHRICHTOCP
|
8.9 | IC50 | 2 | — | |
BYPWTZRGWLOOAC
|
8.9 | IC50 | 2 | — | |
OASUZJWWTNKKNW
|
8.8 | IC50 | 2 | — | |
RXAXXPSLZPTWET
|
8.8 | IC50 | 2 | — | |
ZBPTYYFUGHUNMQ
|
8.8 | IC50 | 2 | — | |
ZPWIFPUPFCEENX
|
8.8 | IC50 | 2 | — | |
ACKBFDXVYCQQDK
|
8.8 | IC50 | 2 | — | |
QDRFBFCKKOITJI
|
8.8 | IC50 | 2 | — | |
BMMZGWDGXPPDEW
|
8.8 | IC50 | 2 | — | |
IRIRGFCFAMOTLN
|
8.8 | IC50 | 2 | — | |
JZUKYILZIUEOPZ
|
8.8 | IC50 | 2 | — | |
KBLQETSGJBJTIR
|
8.8 | IC50 | 2 | — | |
USBMOTXWBABNGC
|
8.8 | IC50 | 2 | — | |
XNVAPQIDSALKTN
|
8.8 | IC50 | 2 | — | |
BLZGGHVIKCCXDY
|
8.8 | IC50 | 2 | — | |
XQRVINZFDOUPSD
|
8.8 | IC50 | 2 | — | |
GAWGUDTUQRRPQK
|
8.7 | IC50 | 2 | — | |
OWWRMDBDEKIWBK
|
8.7 | IC50 | 2 | — | |
WJASKODGMHBDFO
|
8.7 | IC50 | 5 | — | |
AQSSMEORRLJZLU
|
8.7 | Kd | 34 | Yes | |
IRDIFSAZOXFGSK
|
8.7 | IC50 | 2 | — | |
XPASUDUUTHMDBC
|
8.7 | IC50 | 2 | — | |
FHTCHCUICJOIGJ
|
8.7 | IC50 | 7 | — | |
NWZOSSQOJBZGSI
|
8.6 | IC50 | 2 | — | |
RRLYHXUPURJIJM
|
8.6 | IC50 | 2 | — | |
DXVXGQDTEZKMLS
|
8.6 | IC50 | 2 | — | |
JFQUUTOBSZUMCQ
|
8.6 | IC50 | 2 | — | |
XXNVWTNREKGECR
|
8.6 | IC50 | 2 | — | |
LLFCXRYULHMNCG
|
8.6 | IC50 | 2 | — | |
DIDDNVPEZKJYOM
|
8.5 | IC50 | 2 | — | |
WFURCCZQGVBPRV
|
8.5 | IC50 | 2 | — | |
OZMSMXIUMHBELF
|
8.5 | IC50 | 2 | — | |
RORITMKRNLYYLH
|
8.5 | IC50 | 2 | — | |
RYBJAVABBYLDEP
|
8.5 | IC50 | 2 | — | |
SZETXTFRBXNRRT
|
8.5 | IC50 | 2 | — |