Target Details
| UniProt AC | P36897 |
|---|---|
| Gene Symbol | TGFBR1 |
| Protein Name | TGF-beta receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 428
- Clinical molecules 14
- Avg pChEMBL 7.75
KEGG Pathways (23)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Apelin signaling pathway
- Cellular senescence
- Chagas disease
- Chronic myeloid leukemia
- Colorectal cancer
- Cytokine-cytokine receptor interaction
- Diabetic cardiomyopathy
- Endocytosis
- FoxO signaling pathway
- Gastric cancer
- Hepatitis B
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human T-cell leukemia virus 1 infection
- MAPK signaling pathway
- Osteoclast differentiation
- Pancreatic cancer
- Pathways in cancer
- Relaxin signaling pathway
- TGF-beta signaling pathway
- Th17 cell differentiation
Associated Diseases (3)
Active Molecules (428)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RAYASLMMTCQZGM
|
9.7 | IC50 | 2 | — | |
GDGJWSLJIGCBGE
|
9.6 | IC50 | 2 | — | |
WTZAWAYSHRQGOB
|
9.6 | IC50 | 2 | — | |
OFFLEANUVDDEBL
|
9.6 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
9.6 | Kd | 599 | — | |
MGHJYWHFIWPSNB
|
9.5 | IC50 | 2 | — | |
VICAQGVISLDXME
|
9.5 | IC50 | 2 | — | |
DRDNNBDHDQBCMC
|
9.5 | IC50 | 2 | — | |
JFAHUOXKADNXHK
|
9.4 | IC50 | 2 | — | |
IOCHRHMTSUGIPK
|
9.4 | IC50 | 2 | — | |
CHAIHARSRAHKQQ
|
9.4 | IC50 | 2 | — | |
OXAZKHAKYFXQPB
|
9.4 | IC50 | 2 | — | |
MBGUKRYARWDEQD
|
9.3 | IC50 | 2 | — | |
ULMJOBGKUKPBKO
|
9.3 | IC50 | 2 | — | |
HJTMXUSRFLGCTK
|
9.3 | IC50 | 2 | — | |
PCPUDOGTYFUPFV
|
9.3 | IC50 | 2 | — | |
OSXBIOFAAZPBTB
|
9.2 | IC50 | 2 | — | |
KYGGBIHPYVWDIQ
|
9.2 | IC50 | 2 | — | |
OKWIIOORSZALCS
|
9.2 | IC50 | 2 | — | |
DBWYDBLIBRDZNH
|
9.2 | IC50 | 2 | — | |
OCCXAEOXDQXBHG
|
9.2 | IC50 | 2 | — | |
YFMRWYHXGBJCCC
|
9.2 | IC50 | 2 | — | |
JKAPZPMQKNTGJW
|
9.2 | IC50 | 2 | — | |
NHXWKPGFUOSQCJ
|
9.2 | IC50 | 2 | — | |
LXSCQGMBFODPHP
|
9.2 | IC50 | 2 | — | |
BYNUJHIHRYVHIS
|
9.2 | IC50 | 2 | — | |
FOVQNHTXUOXIEW
|
9.2 | IC50 | 2 | — | |
BQEUWLSQIXDQRX
|
9.1 | IC50 | 2 | — | |
XTCDENUICFWZKD
|
9.1 | IC50 | 2 | — | |
JQZQDEAJANBRTM
|
9.1 | IC50 | 2 | — | |
OPHBHEKMLVUZBO
|
9.1 | IC50 | 2 | — | |
LNKMOULIMCFXDG
|
9.1 | IC50 | 2 | — | |
MGCYGWOVPKUJBC
|
9.1 | IC50 | 2 | — | |
RIAWKODQFUGNFD
|
9.1 | IC50 | 2 | — | |
HCZOMSNBQCWQJO
|
9.1 | IC50 | 2 | — | |
YDBNEDDJBRLASN
|
9.1 | IC50 | 2 | — | |
CPUGCQQDYFHDEM
|
9.1 | IC50 | 2 | — | |
FVJODNBTCUGTJZ
|
9.1 | IC50 | 2 | — | |
BGASSDNBKMOKEZ
|
9.1 | IC50 | 2 | — | |
GBOJIFPLPDQYNY
|
9.1 | IC50 | 2 | — | |
WIBYDWSNIHNEPL
|
9.1 | IC50 | 2 | — | |
OWAWLQLFAIHPQT
|
9.1 | IC50 | 2 | — | |
RWIZWKXJKLBCDI
|
9.1 | IC50 | 2 | — | |
LILHDFQTAZTSON
|
9.1 | IC50 | 2 | — | |
TXRZDWUIAYQQJI
|
9.1 | IC50 | 2 | — | |
LDSCHZSRQSLWQV
|
9.0 | IC50 | 2 | — | |
OPGBVTXYOCNCFU
|
9.0 | IC50 | 2 | — | |
BGASSDNBKMOKEZ
|
9.0 | IC50 | 2 | — | |
JGJFSDNRKJRVQG
|
9.0 | IC50 | 2 | — | |
SLMLHNHQKOPWPC
|
9.0 | IC50 | 2 | — |