Target Details
| UniProt AC | P36896 |
|---|---|
| Gene Symbol | ACVR1B |
| Protein Name | Activin receptor type-1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 107
- Clinical molecules 10
- Avg pChEMBL 7.07
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (107)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQWUGDVOUVUTOY
|
7.0 | Kd | 231 | Yes | |
ATSRJSICZUBQJU
|
7.0 | IC50 | 2 | — | |
BVWNOAMYVMKTGC
|
7.0 | IC50 | 3 | — | |
ZBOSAPQCJDMZCV
|
7.0 | IC50 | 6 | — | |
CDOVNWNANFFLFJ
|
6.9 | IC50 | 10 | — | |
PAHLIVNOHVHPBG
|
6.9 | IC50 | 6 | — | |
SRVVCPDKVNJPAH
|
6.9 | IC50 | 2 | — | |
UPBPVAZUFAXUAC
|
6.9 | IC50 | 6 | — | |
OUKYUETWWIPKQR
|
6.8 | Kd | 31 | Yes | |
FHRZBVSUXBSDPP
|
6.8 | IC50 | 2 | — | |
LKZOWZZOQPWIFO
|
6.8 | IC50 | 2 | — | |
FIGRKDLMTBPIFC
|
6.8 | IC50 | 2 | — | |
UEFCSGDOOJJXTN
|
6.8 | IC50 | 46 | — | |
XMGRGPZCVNKAOK
|
6.8 | IC50 | 2 | — | |
XMGRGPZCVNKAOK
|
6.8 | IC50 | 2 | — | |
XBGWAKUQSRNWMA
|
6.7 | IC50 | 4 | — | |
FHYUGAJXYORMHI
|
6.7 | Kd | 7 | — | |
UQEFQNWFVJXGDE
|
6.7 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
6.7 | Kd | 112 | — | |
IVRXNBXKWIJUQB
|
6.7 | IC50 | 10 | — | |
QNABDSWBQJKBHK
|
6.7 | IC50 | 45 | — | |
AQPVZDUZQVWOEP
|
6.7 | IC50 | 3 | — | |
CKLULXBYHFYPHR
|
6.6 | IC50 | 2 | — | |
ROCFHKYAFOQDHC
|
6.6 | IC50 | 5 | — | |
YPTIRJISDXITNF
|
6.6 | IC50 | 3 | — | |
BZXHYPDAQAEAKY
|
6.5 | IC50 | 5 | — | |
SZVLDZCYMADNPG
|
6.5 | IC50 | 3 | — | |
ZBNZXTGUTAYRHI
|
6.5 | Kd | 102 | Yes | |
XYIZJZFZXCURDK
|
6.5 | IC50 | 5 | — | |
DEVVDJCRLJUDBW
|
6.4 | IC50 | 2 | — | |
UBTPOMHEYRBEHT
|
6.4 | IC50 | 5 | — | |
LCVIRAZGMYMNNT
|
6.4 | Kd | 20 | — | |
WFZZPLAPENBNIY
|
6.3 | IC50 | 3 | — | |
KVDFCDPSKGACEZ
|
6.3 | IC50 | 4 | — | |
DSJFEZATROEIML
|
6.3 | IC50 | 2 | — | |
LVEUPFUJRKZPEN
|
6.3 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
6.3 | Kd | 64 | Yes | |
JROFGZPOBKIAEW
|
6.3 | Kd | 10 | — | |
SHWKNOUREYUNBF
|
6.2 | IC50 | 6 | — | |
AGMGRCAUAZCHPG
|
6.2 | IC50 | 5 | — | |
BFSMGDJOXZAERB
|
6.2 | Kd | 33 | — | |
RUBWYYYEDDAWLB
|
6.2 | IC50 | 5 | — | |
NYYYLFUSXWJOML
|
6.2 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
6.2 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.2 | Kd | 213 | — | |
CNEUJSQUCXSRDD
|
6.2 | Kd | 7 | — | |
LYADGAGFYYXXIO
|
6.1 | IC50 | 82 | — | |
JUUFLLKHNYWHKP
|
6.1 | Kd | 12 | — | |
IEJPGJXAWUJROQ
|
6.1 | IC50 | 5 | — | |
LOLPPWBBNUVNQZ
|
6.1 | Kd | 97 | Yes |