Target Details
| UniProt AC | P36894 |
|---|---|
| Gene Symbol | BMPR1A |
| Protein Name | Bone morphogenetic protein receptor type-1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 114
- Clinical molecules 7
- Avg pChEMBL 6.55
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (114)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HGJYCMLNAQLZFL
|
6.0 | IC50 | 3 | — | |
MPUAEAFJNJDWLV
|
6.0 | IC50 | 3 | — | |
SMMLJZCTRMSMMI
|
6.0 | IC50 | 3 | — | |
ZNGBDCDUILRYET
|
6.0 | IC50 | 3 | — | |
BBWFHMVFMVFXJP
|
6.0 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
6.0 | Kd | 289 | Yes | |
GAIBPGQSYNAFNN
|
6.0 | IC50 | 3 | — | |
MOTRKLJWPDOTBN
|
6.0 | IC50 | 3 | — | |
BBWFHMVFMVFXJP
|
6.0 | IC50 | 3 | — | |
GAIBPGQSYNAFNN
|
6.0 | IC50 | 3 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KRLRRZRTVIVROZ
|
6.0 | IC50 | 3 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |