Target Details
| UniProt AC | P36894 |
|---|---|
| Gene Symbol | BMPR1A |
| Protein Name | Bone morphogenetic protein receptor type-1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 114
- Clinical molecules 7
- Avg pChEMBL 6.55
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (114)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JTVBXQAYBIJXRP
|
6.5 | Kd | 20 | — | |
WIMYXIDFXOAJPL
|
6.5 | IC50 | 3 | — | |
ZBOSAPQCJDMZCV
|
6.5 | IC50 | 6 | — | |
YTUZELSDHUVEFM
|
6.5 | IC50 | 4 | — | |
GIAGHNVPQYZDIK
|
6.4 | IC50 | 3 | — | |
JDAFKLSYNCTYHC
|
6.4 | IC50 | 3 | — | |
SCHRCCHASZMVAB
|
6.4 | IC50 | 7 | — | |
LOLPPWBBNUVNQZ
|
6.4 | Kd | 97 | Yes | |
FYPPBYUPMODRPA
|
6.4 | IC50 | 4 | — | |
WSNLCMQIUFLQBS
|
6.4 | IC50 | 3 | — | |
AWERICKZHUFDGO
|
6.4 | IC50 | 3 | — | |
FFLJVBPCONQSQW
|
6.4 | IC50 | 8 | — | |
RKBYYWVZFBATHQ
|
6.4 | IC50 | 12 | — | |
BKJSJLXWFRXVNO
|
6.3 | IC50 | 2 | — | |
ICKRRSVRNGVVPJ
|
6.3 | IC50 | 2 | — | |
QKDBOJCTMDJVMH
|
6.3 | IC50 | 4 | — | |
NTLWKKILBCETHV
|
6.3 | IC50 | 4 | — | |
FZJGVHATMCAPLO
|
6.3 | IC50 | 5 | — | |
MEDZXCCPJFWNLJ
|
6.3 | IC50 | 3 | — | |
OVNAOUBDNBHVCI
|
6.3 | IC50 | 5 | — | |
LJUBHCPBQBKBHM
|
6.3 | IC50 | 5 | — | |
MEDZXCCPJFWNLJ
|
6.3 | IC50 | 3 | — | |
PDSJQPLUVYRPDN
|
6.3 | IC50 | 3 | — | |
ZCCPLJOKGAACRT
|
6.3 | Kd | 599 | — | |
BBDGBGOVJPEFBT
|
6.3 | IC50 | 6 | — | |
SOXBHNNRUKELLI
|
6.3 | IC50 | 3 | — | |
WOAXRKYXUKTLEM
|
6.3 | IC50 | 7 | — | |
PRKWSDOLROTYLX
|
6.2 | IC50 | 3 | — | |
HZMKNGJNPOBODV
|
6.2 | IC50 | 4 | — | |
UOAHJPVGHFVHGE
|
6.2 | IC50 | 4 | — | |
VUEWHTWKZUEQMF
|
6.2 | IC50 | 4 | — | |
GGDVEPRDLUWBFD
|
6.2 | IC50 | 4 | — | |
UOTRHTRIIAWPIM
|
6.2 | IC50 | 3 | — | |
DHQCKBUTDYGTKB
|
6.2 | IC50 | 3 | — | |
DPDIGSURNQRYQS
|
6.1 | IC50 | 3 | — | |
JXPPULPLYFLFJI
|
6.1 | IC50 | 3 | — | |
ABEPADPRAQLNSN
|
6.1 | IC50 | 3 | — | |
FCKKBQZIGVYODN
|
6.1 | IC50 | 4 | — | |
YFNWWNRZJGMDBR
|
6.1 | Kd | 35 | — | |
GPLMXGSESNBQQL
|
6.1 | IC50 | 3 | — | |
LLFCXRYULHMNCG
|
6.1 | IC50 | 2 | — | |
TUFWPHNCGNFLJQ
|
6.1 | IC50 | 3 | — | |
GNDTWZQOAXPKCV
|
6.1 | IC50 | 3 | — | |
UKJHXNZUFMVJFI
|
6.1 | IC50 | 3 | — | |
KIUMBIWMXBUHDW
|
6.0 | IC50 | 3 | — | |
KPRPFTOLWQQUAV
|
6.0 | IC50 | 3 | — | |
MKKQYAXMQPGYNY
|
6.0 | IC50 | 3 | — | |
MXDCACLUETVZNL
|
6.0 | IC50 | 8 | — | |
RQXROVVCXFAAOM
|
6.0 | IC50 | 3 | — | |
SGIKWGLEUPAMLM
|
6.0 | IC50 | 3 | — |