Target Details
| UniProt AC | P36894 |
|---|---|
| Gene Symbol | BMPR1A |
| Protein Name | Bone morphogenetic protein receptor type-1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 114
- Clinical molecules 7
- Avg pChEMBL 6.55
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (114)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WJASKODGMHBDFO
|
8.6 | IC50 | 5 | — | |
FAOGJKJCGFIFLI
|
8.2 | IC50 | 6 | — | |
SHWKNOUREYUNBF
|
8.1 | IC50 | 6 | — | |
WCDLCPLAAKUJNY
|
8.0 | IC50 | 8 | — | |
CDOVNWNANFFLFJ
|
7.7 | IC50 | 10 | — | |
MQFUFNHTCJRLKW
|
7.5 | IC50 | 6 | — | |
UPBPVAZUFAXUAC
|
7.5 | IC50 | 6 | — | |
CJLMANFTWLNAKC
|
7.5 | IC50 | 5 | — | |
IIYOBXCNRFSCBH
|
7.4 | IC50 | 8 | — | |
PAHLIVNOHVHPBG
|
7.3 | IC50 | 6 | — | |
WMTXIPYJYDISKM
|
7.3 | IC50 | 8 | — | |
FHTCHCUICJOIGJ
|
7.2 | IC50 | 7 | — | |
LYZXDNCSIHIAMI
|
7.2 | IC50 | 3 | — | |
OUKYUETWWIPKQR
|
7.2 | Kd | 31 | Yes | |
ROCFHKYAFOQDHC
|
7.2 | IC50 | 5 | — | |
MFAQYJIYDMLAIM
|
7.2 | Kd | 130 | Yes | |
KVLSZJPFQDRDPI
|
7.2 | IC50 | 4 | — | |
XIFIYBGPRFRYNP
|
7.1 | IC50 | 4 | — | |
OVXMCCQKIOSDGE
|
7.0 | IC50 | 3 | — | |
XHBVYDAKJHETMP
|
7.0 | IC50 | 24 | Yes | |
RZYYJEYQNNJBMD
|
6.9 | IC50 | 3 | — | |
WJSYQJFCHPTVCI
|
6.9 | IC50 | 3 | — | |
IEJPGJXAWUJROQ
|
6.9 | IC50 | 5 | — | |
UAHBMBZHEHEEAW
|
6.8 | IC50 | 4 | — | |
ZOMQASFZVQEKHR
|
6.8 | IC50 | 3 | — | |
AJRCHNXNYNADRQ
|
6.8 | IC50 | 3 | — | |
SRIVDECCESIDAQ
|
6.8 | IC50 | 3 | — | |
RIWTUJFFSTVYPW
|
6.8 | IC50 | 6 | — | |
DUGKWSLUPDXHDO
|
6.8 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
VAARYSWULJUGST
|
6.8 | Kd | 119 | Yes | |
BLKUTJODYRMUJL
|
6.7 | IC50 | 4 | — | |
QQYOZULVMVWDFQ
|
6.7 | IC50 | 3 | — | |
XJRNYUDHNXZYCF
|
6.7 | IC50 | 3 | — | |
XQLHGVZYEZLJEG
|
6.7 | IC50 | 3 | — | |
OBLCGNSTBZOGIQ
|
6.7 | IC50 | 3 | — | |
ALKJNCZNEOTEMP
|
6.7 | Kd | 55 | — | |
WTMROIBZVGJXRP
|
6.7 | IC50 | 4 | — | |
XYIZJZFZXCURDK
|
6.7 | IC50 | 5 | — | |
UTCHZVUDAGSGMY
|
6.7 | IC50 | 3 | — | |
KIAKJNRDKPGTQR
|
6.6 | IC50 | 6 | — | |
ODVUZZFWFOPOAH
|
6.6 | IC50 | 5 | — | |
JDYMCSKANXEKMK
|
6.6 | IC50 | 3 | — | |
QCXBJMRMYRQRCV
|
6.6 | IC50 | 4 | — | |
IFSNOUHZJMGMOD
|
6.5 | IC50 | 4 | — | |
RIGIHWPKCOSNDD
|
6.5 | IC50 | 3 | — | |
UXVFRKCJRULCNV
|
6.5 | IC50 | 4 | — | |
HIWHLPKRUZGHRR
|
6.5 | IC50 | 4 | — | |
GGQCWUKLPMFTDA
|
6.5 | IC50 | 5 | — | |
PVDWNOWJXDXMDH
|
6.5 | IC50 | 5 | — |