Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UZEICMNTLHFXNT
|
8.5 | IC50 | 2 | — | |
DVPCNIKFABUUTG
|
8.5 | Kd | 2 | — | |
MQQQNGBBTVKGQZ
|
8.5 | IC50 | 4 | — | |
YHTAHGYPUILKPD
|
8.5 | IC50 | 2 | — | |
ZFBBKOBKYNRTOS
|
8.5 | IC50 | 4 | — | |
HSJCSHDUINVROZ
|
8.5 | IC50 | 4 | — | |
MWXLURJNASFGGM
|
8.5 | IC50 | 5 | — | |
VXGBFWNTVZKGOT
|
8.5 | IC50 | 3 | — | |
PIQCTGMSNWUMAF
|
8.4 | Kd | 137 | Yes | |
VZOFLHLWMKWZHW
|
8.4 | IC50 | 4 | — | |
YUOGCICHWDJBLS
|
8.4 | IC50 | 2 | — | |
GTDOWKUTGWWIFA
|
8.4 | IC50 | 3 | — | |
CDPXZDPKRHLKCH
|
8.4 | IC50 | 4 | — | |
DGHMFYHSNOIJHK
|
8.4 | IC50 | 2 | — | |
NLXWFBBYANWXPR
|
8.4 | IC50 | 4 | — | |
SUXYGJZMCWKJJI
|
8.4 | IC50 | 26 | Yes | |
UGZGQNGZCRYGKF
|
8.4 | IC50 | 3 | — | |
WDVWNWIIOYPZAE
|
8.4 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
8.4 | Kd | 165 | Yes | |
MBOBSHMPDSNBHM
|
8.4 | IC50 | 2 | — | |
WORRXRIVSMTSEB
|
8.4 | IC50 | 4 | — | |
AKWLDQDWZNJYKL
|
8.4 | IC50 | 14 | — | |
APUCFXHENVUXCY
|
8.4 | Ki | 15 | — | |
AXXUSLKWELMYSS
|
8.4 | IC50 | 3 | — | |
BGYVWFZMYBWCNY
|
8.4 | Ki | 30 | — | |
CPJULNXNBQMSHF
|
8.4 | IC50 | 3 | — | |
DGLXOJMLPNCUDE
|
8.4 | IC50 | 7 | Yes | |
DLYHIJZSZUMFEL
|
8.4 | IC50 | 5 | Yes | |
DVJRDKAXQCFWKO
|
8.4 | IC50 | 2 | — | |
FUNGTOAZDDISQB
|
8.4 | IC50 | 4 | Yes | |
GEGCXGMFUYJULA
|
8.4 | IC50 | 30 | Yes | |
GSQNTGGWLBUZMI
|
8.4 | IC50 | 3 | — | |
HMAFXPLOLABOEY
|
8.4 | IC50 | 3 | — | |
IKENQUDOTQBCJH
|
8.4 | Kd | 18 | — | |
JPWGMNSPCZZICA
|
8.4 | IC50 | 4 | — | |
LSLPDHNUWRDOGC
|
8.4 | Ki | 25 | — | |
LVECPYVAIBNSRV
|
8.4 | Ki | 33 | — | |
MMCWBZCSGNCOMQ
|
8.4 | IC50 | 5 | Yes | |
MULNSLQVKKUPJN
|
8.4 | Ki | 41 | — | |
MVJMMLFMPWITEJ
|
8.4 | Ki | 110 | — | |
NGBFROQDGZCMCE
|
8.4 | IC50 | 3 | — | |
NZCHGHMPHKCWLR
|
8.4 | IC50 | 6 | — | |
OBSFXHDOLBYWRJ
|
8.4 | IC50 | 7 | Yes | |
OHUNADGDEWQCLI
|
8.4 | IC50 | 2 | — | |
PJSBFZAYJQMORO
|
8.4 | Ki | 11 | — | |
PPPOUAQYRUUFNJ
|
8.4 | IC50 | 3 | — | |
QJYWNLGATZHNCX
|
8.4 | IC50 | 4 | — | |
RIUZPIBUSOHUKF
|
8.4 | Ki | 23 | — | |
SXSIVJXOXSHKPK
|
8.4 | IC50 | 5 | Yes | |
UFSGCADQVRKELP
|
8.4 | IC50 | 3 | — |