Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ROIWAJLBBPZORU
|
8.5 | IC50 | 4 | — | |
WZSUDZDKYJWJPS
|
8.5 | IC50 | 4 | — | |
BBJHTTNJKZUZCD
|
8.5 | IC50 | 4 | — | |
DUHXDQPGUINDGD
|
8.5 | IC50 | 3 | — | |
DYQYODJNEBRPRK
|
8.5 | IC50 | 4 | — | |
DYSDUQPAIATDAA
|
8.5 | IC50 | 5 | Yes | |
HGLWPJISHDLCTE
|
8.5 | IC50 | 7 | — | |
HHKOKFHTWVYTJK
|
8.5 | IC50 | 4 | — | |
HMRCNHLZGISKIM
|
8.5 | IC50 | 4 | Yes | |
KAAPXWSYROPAEL
|
8.5 | IC50 | 4 | — | |
LFOWPAZJQIZNHI
|
8.5 | IC50 | 4 | — | |
LKMNVWCDUCOIDP
|
8.5 | IC50 | 2 | — | |
LMEANLPGOCWAMD
|
8.5 | IC50 | 3 | — | |
PPPOUAQYRUUFNJ
|
8.5 | IC50 | 4 | — | |
PTRVZEMPNWFZEI
|
8.5 | IC50 | 4 | — | |
QPNALTDCQOTWLI
|
8.5 | IC50 | 4 | Yes | |
RBARWKMXQSXULQ
|
8.5 | IC50 | 3 | — | |
SBYAVEOYFSHPBT
|
8.5 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
8.5 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
8.5 | Kd | 289 | Yes | |
VCQXPLQAUTUUTC
|
8.5 | IC50 | 3 | — | |
WOINYYVWAXSXMQ
|
8.5 | IC50 | 4 | Yes | |
XCHZMPYWMULFBJ
|
8.5 | IC50 | 4 | Yes | |
XTKIFGMBONJHTF
|
8.5 | IC50 | 4 | Yes | |
LFOWPAZJQIZNHI
|
8.5 | IC50 | 4 | — | |
MAHJDNICCJZVKW
|
8.5 | IC50 | 4 | — | |
NATOVXPHBATGAZ
|
8.5 | IC50 | 2 | — | |
RATPJUQSJPMXQH
|
8.5 | IC50 | 4 | — | |
UCRFEDKYGLHWFM
|
8.5 | IC50 | 2 | — | |
XLRGWOQAKMIFSL
|
8.5 | IC50 | 2 | — | |
FGSVLADZCDNNOC
|
8.5 | Ki | 11 | — | |
GCYXEGSPUDSZJY
|
8.5 | Ki | 82 | — | |
GSXRCPJTNIGKSZ
|
8.5 | Ki | 43 | — | |
JVAUXOQNQAAUBJ
|
8.5 | IC50 | 3 | — | |
KOHNRDPXFDZZJF
|
8.5 | Ki | 31 | — | |
RKLGMDOZEOTQEM
|
8.5 | Ki | 12 | — | |
RYAVJHIPOWNWDE
|
8.5 | Ki | 38 | — | |
WSRSUSKJBOADHJ
|
8.5 | IC50 | 3 | — | |
XVFMIEBCFYSYBS
|
8.5 | IC50 | 2 | — | |
ZXLFIHLBHMLHFJ
|
8.5 | Ki | 31 | — | |
GWILJQBMYLXBHZ
|
8.5 | Kd | 4 | — | |
IADRGGYOCXDICI
|
8.5 | IC50 | 4 | — | |
RXKJTHMWVQQQRO
|
8.5 | IC50 | 4 | — | |
UMHCVDDSESEXLS
|
8.5 | IC50 | 4 | — | |
YJRPVMCKBPJNKR
|
8.5 | IC50 | 2 | — | |
YQUHLIQEGXFNCX
|
8.5 | IC50 | 2 | — | |
BPKUEQDPPXTOSG
|
8.5 | IC50 | 4 | — | |
CKRMOFCKEANQCR
|
8.5 | IC50 | 4 | — | |
JQNUCFXJVXYPNW
|
8.5 | IC50 | 2 | — | |
OKIKSBCVNZBYGX
|
8.5 | IC50 | 5 | — |