Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKBFHTIUXUCYRQ
|
8.7 | IC50 | 8 | — | |
WTWMNNKZEVJCBK
|
8.7 | IC50 | 5 | — | |
YBZJHECNTDHGQY
|
8.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.7 | Kd | 213 | — | |
BFAFTEXTXVWPSX
|
8.6 | IC50 | 5 | Yes | |
MUIPWSHBCRIWKJ
|
8.6 | IC50 | 4 | — | |
QQWUCWPOJLZHJB
|
8.6 | IC50 | 3 | — | |
SGTSFIPSFBYYSH
|
8.6 | IC50 | 4 | — | |
VTWWRKFUHCSCEW
|
8.6 | Kd | 19 | — | |
YQUHLIQEGXFNCX
|
8.6 | IC50 | 2 | — | |
WLTXIECTWSMSQB
|
8.6 | IC50 | 2 | — | |
BLQYVHBZHAISJM
|
8.6 | IC50 | 21 | Yes | |
BLQYVHBZHAISJM
|
8.6 | IC50 | 54 | — | |
GOTODHLHVSBWDG
|
8.6 | Kd | 2 | — | |
RTZPWZZLLAHMAA
|
8.6 | IC50 | 4 | — | |
JBBBYMPMAJVCSI
|
8.6 | IC50 | 3 | Yes | |
DKZQQJXYLNUWFT
|
8.6 | IC50 | 4 | — | |
GDEJPGKNPRJNGE
|
8.6 | Ki | 6 | — | |
JKQBDGDSVVQSGS
|
8.6 | IC50 | 2 | — | |
KGSRYTUWXUESJK
|
8.6 | IC50 | 7 | — | |
NSLJACGCOKVYOC
|
8.6 | IC50 | 4 | — | |
RPDVCUCXMGWTFA
|
8.6 | Ki | 10 | — | |
SFPWNTQWFFNJIH
|
8.6 | Ki | 48 | — | |
ITRYMWSQXXWWJF
|
8.6 | IC50 | 4 | — | |
ORIMXTQTVHCGIW
|
8.6 | IC50 | 4 | — | |
OVSVIUOGHPWXNH
|
8.6 | IC50 | 6 | — | |
VUZLNWIIHACTEC
|
8.6 | IC50 | 4 | — | |
WERQRDFKILOXSK
|
8.6 | IC50 | 4 | — | |
WOVFEULIRSIJJU
|
8.6 | IC50 | 4 | — | |
XLRGWOQAKMIFSL
|
8.6 | IC50 | 2 | — | |
AAUNIEBMIUGNTA
|
8.6 | IC50 | 4 | — | |
CDKUUJPCCTYLGH
|
8.6 | IC50 | 2 | — | |
HRCFERVVUBEPAE
|
8.6 | IC50 | 2 | — | |
PHLVHKVYPBUWOL
|
8.6 | IC50 | 7 | — | |
ULNQWYGVWVDLPK
|
8.6 | IC50 | 2 | — | |
VOEBMPAZQQYYGC
|
8.6 | IC50 | 5 | Yes | |
XTXMJKTXFRAXRP
|
8.6 | IC50 | 2 | — | |
ZPOKSLXILOTPCR
|
8.6 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
8.6 | Kd | 599 | — | |
FJWZASZEWLWFRB
|
8.6 | IC50 | 4 | — | |
HBQLAXMLLMAJCM
|
8.6 | IC50 | 4 | — | |
IEXXROGGKUBLPS
|
8.6 | IC50 | 4 | — | |
IGIRIPQQEQZJIY
|
8.6 | Ki | 8 | — | |
IZDBEJJRNUSRIU
|
8.6 | IC50 | 3 | — | |
QBBXSRZGLKRAMO
|
8.6 | IC50 | 4 | — | |
UMJNEGIWFHRTLO
|
8.6 | IC50 | 4 | — | |
VSNJCPXJAHKLRS
|
8.6 | Ki | 7 | Yes | |
AZVXPGDWKUCGLO
|
8.5 | IC50 | 2 | — | |
LSEAQLOYCHTEOK
|
8.5 | IC50 | 10 | — | |
POFRIXOEJZMCHH
|
8.5 | IC50 | 2 | — |