Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.7 | IC50 | 408 | — | |
AEOFEGDYORZHFE
|
8.7 | IC50 | 4 | — | |
AGIHELYBRFIVHZ
|
8.7 | IC50 | 4 | — | |
AZIKDQBYCZVPSU
|
8.7 | IC50 | 3 | — | |
BXVHRRLJGZKCBN
|
8.7 | IC50 | 2 | — | |
CWFMWJSSAAOUBO
|
8.7 | IC50 | 4 | — | |
FGYMKXFFIWSCGZ
|
8.7 | IC50 | 4 | — | |
FQYLJBVSYHZWLT
|
8.7 | IC50 | 35 | Yes | |
HHVUHFYJIYORJI
|
8.7 | IC50 | 3 | — | |
HWEBFAZCYKVEJD
|
8.7 | IC50 | 5 | — | |
HXYSWTZEQZNVDR
|
8.7 | IC50 | 3 | — | |
IAURWWSIIMOBHU
|
8.7 | IC50 | 4 | — | |
JGFZPZGREYNUPH
|
8.7 | IC50 | 5 | Yes | |
KMDUVZLDXOHFPQ
|
8.7 | IC50 | 4 | — | |
KXMZDGSRSGHMMK
|
8.7 | IC50 | 14 | — | |
LYHXSDWIWVVZPB
|
8.7 | IC50 | 6 | Yes | |
MENVZXUPTOFKRC
|
8.7 | IC50 | 3 | — | |
PKAXKMPZRBQIOO
|
8.7 | IC50 | 3 | — | |
PTVPBWWDGZSEAF
|
8.7 | Ki | 63 | — | |
QONPPIZSNSSCSK
|
8.7 | IC50 | 45 | Yes | |
REZSMOYMCKDNEU
|
8.7 | IC50 | 3 | — | |
RKILQDBEPHSTGP
|
8.7 | IC50 | 3 | — | |
RKILQDBEPHSTGP
|
8.7 | IC50 | 4 | — | |
RROPCZKHYUPTGO
|
8.7 | IC50 | 3 | — | |
SXOGNSSKJOUDNZ
|
8.7 | IC50 | 4 | — | |
UKUVHVSOTZPZBW
|
8.7 | IC50 | 4 | — | |
UOOZSMNSBYVUGZ
|
8.7 | Ki | 32 | — | |
UWDBNTXEKYRMSG
|
8.7 | Ki | 26 | — | |
VPDYUDURNXPNMA
|
8.7 | IC50 | 5 | Yes | |
WVXNSAVVKYZVOE
|
8.7 | IC50 | 92 | — | |
XLFYOIVELARSKP
|
8.7 | Ki | 33 | — | |
XYXLUJQBBIBJFV
|
8.7 | Ki | 36 | — | |
ZVVIKPIHXSNXJY
|
8.7 | IC50 | 4 | Yes | |
ZZXOJMDHTLVJPY
|
8.7 | IC50 | 2 | — | |
AILRADAXUVEEIR
|
8.7 | IC50 | 75 | — | |
FZBVNCFBCNXULH
|
8.7 | IC50 | 18 | — | |
GFXJPWQHPZNCGC
|
8.7 | IC50 | 3 | — | |
HYDSSXBBNYALNP
|
8.7 | IC50 | 5 | — | |
MIYIUVBGBPRNLG
|
8.7 | IC50 | 4 | — | |
RBMXNQRKVSGKHT
|
8.7 | IC50 | 2 | — | |
ULHLSSWDQFLSBL
|
8.7 | IC50 | 6 | — | |
XGIIMGRAMUXNFL
|
8.7 | IC50 | 4 | — | |
HBQMROYUNHRFSB
|
8.7 | IC50 | 5 | — | |
HFSWCNDZVPIIOF
|
8.7 | IC50 | 8 | — | |
KDBWIIMYOYEZDH
|
8.7 | IC50 | 4 | — | |
NBSJZWFDNFWQDN
|
8.7 | IC50 | 29 | — | |
NDWOEUVAOGUXGP
|
8.7 | IC50 | 4 | — | |
NVHUKBRGAIBVPK
|
8.7 | IC50 | 4 | — | |
OCDYJTRAVKONSS
|
8.7 | Kd | 3 | — | |
SINLAAVSJWFXNK
|
8.7 | IC50 | 4 | — |