Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KRRYGFBABIBCHR
|
8.9 | IC50 | 3 | — | |
PIHKTGDJUXUJMJ
|
8.9 | IC50 | 4 | — | |
VBQONCXEWJGAOC
|
8.9 | IC50 | 3 | — | |
FLEDZRUQPMPOFA
|
8.8 | IC50 | 4 | — | |
MPFWQMHHDIWYNG
|
8.8 | IC50 | 2 | — | |
NNAMXKXTCQOZGS
|
8.8 | IC50 | 5 | Yes | |
BBUVDDPUURMFOX
|
8.8 | IC50 | 3 | — | |
FVXFEJBGHYVGML
|
8.8 | Kd | 2 | — | |
JZCBGMAKTMOCFP
|
8.8 | IC50 | 4 | Yes | |
LPWSVHUTHUTIIH
|
8.8 | IC50 | 2 | — | |
MAIZEWVIGRBICN
|
8.8 | IC50 | 4 | — | |
QDCNDOVOAIZYTL
|
8.8 | IC50 | 4 | — | |
QDCNDOVOAIZYTL
|
8.8 | IC50 | 4 | — | |
SEJGTFPOEJWEGG
|
8.8 | Kd | 149 | — | |
UYDMDSBIXKYMQD
|
8.8 | IC50 | 5 | — | |
VNPYBQLMWOYRMR
|
8.8 | IC50 | 4 | — | |
RLVKBWCJGUWUHI
|
8.8 | IC50 | 2 | — | |
UDVJBRYBBSVDDS
|
8.8 | IC50 | 14 | — | |
WKRSQWJVMBRBPZ
|
8.8 | IC50 | 3 | — | |
YFLNJIAXYKROBA
|
8.8 | IC50 | 3 | — | |
BWLVWHQFWOPSOP
|
8.8 | IC50 | 4 | — | |
DLJHLQKPFJJSLK
|
8.8 | IC50 | 2 | — | |
FDVSOQRNTAPCHB
|
8.8 | Ki | 40 | — | |
GWMATETWMAQOFL
|
8.8 | Ki | 36 | — | |
KROLCVQARUUHNV
|
8.8 | Ki | 12 | — | |
LHVFNERWJYBEJN
|
8.8 | Kd | 7 | — | |
MFMXAWQGPQXDRJ
|
8.8 | Ki | 27 | — | |
MLIFNJABMANKEU
|
8.8 | IC50 | 9 | Yes | |
OEUMLQMTMOCCGW
|
8.8 | Kd | 6 | — | |
QKPLUKMJEKRAJD
|
8.8 | Ki | 30 | Yes | |
ULHGAQSVFPOUDY
|
8.8 | Ki | 43 | — | |
UTQPKPHUIMHAAN
|
8.8 | Ki | 22 | — | |
VEFDEIILCRXHNC
|
8.8 | IC50 | 4 | — | |
VUVZPZAXDNURQR
|
8.8 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
8.8 | Ki | 66 | — | |
YQUHLIQEGXFNCX
|
8.8 | IC50 | 2 | — | |
ZQQVWTACALNOAJ
|
8.8 | Ki | 11 | — | |
QYMKGQPTZIRPMA
|
8.8 | IC50 | 2 | — | |
CREINZJAYXIGBI
|
8.8 | IC50 | 4 | — | |
ZTAGFSQIVLXCQE
|
8.8 | IC50 | 2 | — | |
AJLUXNJECIAQBR
|
8.7 | IC50 | 4 | — | |
CMWZJGXVESUMJY
|
8.7 | IC50 | 2 | — | |
PRIMAMTZCAWUCI
|
8.7 | IC50 | 2 | — | |
UGEJLCNSVIVALC
|
8.7 | IC50 | 41 | — | |
LYADGAGFYYXXIO
|
8.7 | IC50 | 82 | — | |
OQOSJDFXPZMLPT
|
8.7 | IC50 | 2 | — | |
QNSYKQNSCIEOLI
|
8.7 | IC50 | 5 | Yes | |
RMLWTYYGKGDCFZ
|
8.7 | IC50 | 4 | — | |
UEKBKVAQJQTBGW
|
8.7 | IC50 | 3 | — | |
ADLPKFFMGIJZIM
|
8.7 | IC50 | 44 | — |