Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MMKIEBBLOVSLAS
|
9.0 | IC50 | 3 | — | |
NQZRHTLUKLOASK
|
9.0 | IC50 | 3 | — | |
NSKFXNDKPCVDIN
|
9.0 | Ki | 12 | — | |
NYFSAYXCSAIWGI
|
9.0 | IC50 | 3 | — | |
OOQJIJYKWXLQNC
|
9.0 | IC50 | 16 | Yes | |
OPJBZLDDGJGVCQ
|
9.0 | IC50 | 5 | — | |
QDOBTYVGPGFRCM
|
9.0 | Ki | 11 | — | |
QEVGJXHJXPXEJA
|
9.0 | IC50 | 4 | — | |
UAIANIHUMMKHJR
|
9.0 | IC50 | 3 | — | |
UBKAKYFRDGQVJG
|
9.0 | IC50 | 3 | — | |
ZPXYYHKOOQSKHV
|
9.0 | IC50 | 4 | — | |
LHDKPFSHXFFALR
|
9.0 | IC50 | 7 | — | |
NMWURSLYBLOJKP
|
9.0 | IC50 | 3 | — | |
QOIKDVCHQYXCQL
|
9.0 | IC50 | 2 | — | |
AVQBNZOTTBHSCI
|
9.0 | IC50 | 4 | — | |
UODZHAZSVRMPND
|
9.0 | IC50 | 2 | — | |
YEGSATWQBXVWBX
|
9.0 | IC50 | 6 | — | |
IQZVWRXRHZPRBO
|
8.9 | IC50 | 2 | — | |
NXCNMBDRRSLYBU
|
8.9 | IC50 | 2 | — | |
IXULLLZCNUKGBJ
|
8.9 | IC50 | 6 | — | |
AYLQSRFNFBZNQA
|
8.9 | IC50 | 2 | — | |
CPQMLGLUULWKDX
|
8.9 | IC50 | 4 | Yes | |
DCFNMFYAKVXCLN
|
8.9 | IC50 | 4 | — | |
LBEJYFVJIPQSNX
|
8.9 | IC50 | 4 | — | |
PSABAQPTDYJLPZ
|
8.9 | Kd | 2 | — | |
SZFYZDIPRMLBDC
|
8.9 | Kd | 9 | — | |
BRTHUECZMVKNMQ
|
8.9 | IC50 | 7 | — | |
JEZXMQDUAGEGLR
|
8.9 | IC50 | 2 | — | |
MBDALTHTQIMRAH
|
8.9 | IC50 | 2 | — | |
DZSUJUOJJJCWGG
|
8.9 | IC50 | 55 | Yes | |
KOSUFZUQHXDTAI
|
8.9 | IC50 | 5 | — | |
MCCCQFAOMZMZKE
|
8.9 | Ki | 52 | — | |
PLHUMPJXRHMFFR
|
8.9 | Ki | 28 | — | |
RWEHAHIEUDLKGT
|
8.9 | Ki | 33 | — | |
SQOLAIUZCKYPCQ
|
8.9 | IC50 | 2 | — | |
UXQLMVSZSYZFID
|
8.9 | Ki | 12 | — | |
ZCCJKVBTHCOISJ
|
8.9 | Ki | 46 | — | |
FEXRSRXFBIRFMY
|
8.9 | IC50 | 4 | — | |
HTMNAROLUQALML
|
8.9 | IC50 | 4 | — | |
MJSHVHLADKXCML
|
8.9 | IC50 | 4 | — | |
OBFGRWOUNPRHNH
|
8.9 | IC50 | 6 | — | |
OEJRGRXZSULSGO
|
8.9 | IC50 | 2 | — | |
OYUDNKFIGXAIRZ
|
8.9 | Ki | 16 | Yes | |
UIKRXGNEQUHBIX
|
8.9 | IC50 | 4 | — | |
WPHKIQPVPYJNAX
|
8.9 | IC50 | 81 | — | |
WYCSRUVPJUYDGP
|
8.9 | IC50 | 6 | — | |
NNPRQBLRXNNMJV
|
8.9 | IC50 | 5 | — | |
TZKBVRDEOITLRB
|
8.9 | IC50 | 7 | — | |
OIELVFPEYHWMQZ
|
8.9 | IC50 | 2 | — | |
VEPOCTYIFBFDRZ
|
8.9 | IC50 | 4 | — |