Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MJSHVHLADKXCML
|
9.1 | IC50 | 11 | — | |
MXCUSZDSXDTMHC
|
9.1 | IC50 | 3 | — | |
NHFDRBXTEDBWCZ
|
9.1 | Kd | 12 | Yes | |
PEJCGJUJBCLDFV
|
9.1 | Kd | 2 | — | |
QAKMQVCMEPKBHL
|
9.1 | Ki | 11 | — | |
SJMFZIGFOIPNPE
|
9.1 | Ki | 10 | — | |
UZBFFCBUJQNOPY
|
9.1 | IC50 | 3 | — | |
WGQUSQTWZRXHGK
|
9.1 | IC50 | 3 | — | |
XMUWGNAFKPBEAU
|
9.1 | IC50 | 5 | Yes | |
XMWONVHOMANOOY
|
9.1 | IC50 | 3 | — | |
YMEYAMDEQBMREG
|
9.1 | IC50 | 3 | — | |
BLEFJHDCLNVQNS
|
9.1 | IC50 | 3 | — | |
DYNHJHQFHQTFTP
|
9.1 | Kd | 38 | — | |
QDZSPZAGUMSAMI
|
9.1 | IC50 | 2 | — | |
XHCPCYVQXFHJAU
|
9.1 | IC50 | 12 | — | |
AZUGZDWCCRNTDK
|
9.1 | IC50 | 2 | — | |
MJIIYXFGPPGPGB
|
9.1 | IC50 | 5 | — | |
WMWHVTDZNIVNIE
|
9.1 | IC50 | 9 | — | |
YRUDYNCGPZHXRB
|
9.1 | Kd | 6 | — | |
AKLWVZFHNFDHCQ
|
9.1 | IC50 | 3 | — | |
CMKUJKFQBWYWBJ
|
9.1 | IC50 | 3 | — | |
RAOCKIXJWYDYCO
|
9.1 | IC50 | 5 | Yes | |
RGJASBGADDXMBE
|
9.1 | IC50 | 4 | — | |
VGNWKKQVJCEBCJ
|
9.1 | IC50 | 3 | — | |
YBJQFWOWWBZCJS
|
9.1 | Kd | 2 | — | |
SQOLAIUZCKYPCQ
|
9.0 | IC50 | 3 | — | |
NVLFLJAFSQNISZ
|
9.0 | IC50 | 3 | — | |
QXQKUTDAZQEITC
|
9.0 | IC50 | 4 | — | |
GGLRONBKQRZFOT
|
9.0 | IC50 | 3 | — | |
NSSXXNQRAYKGAQ
|
9.0 | IC50 | 2 | — | |
AKBNGGYXMZTHEB
|
9.0 | IC50 | 5 | — | |
BAEPKCSJXVFDDR
|
9.0 | Kd | 2 | — | |
BBUVDDPUURMFOX
|
9.0 | Kd | 4 | — | |
BIKYDWLMTPRSQL
|
9.0 | Ki | 50 | — | |
CLYZLUAUBTXCPL
|
9.0 | IC50 | 7 | — | |
DBXOMQJZSQLQED
|
9.0 | Ki | 12 | — | |
DUOPMZXNVCHSKJ
|
9.0 | IC50 | 3 | — | |
FLXHMSFCIMZSJT
|
9.0 | IC50 | 3 | — | |
FUOKGTYXSNVQIW
|
9.0 | IC50 | 3 | — | |
GEATXDJAPAHPTP
|
9.0 | IC50 | 10 | — | |
HEPDAJRNJBNJAE
|
9.0 | IC50 | 15 | Yes | |
INOASWZOZPQAQM
|
9.0 | IC50 | 5 | — | |
IWAWFGKTGNXQLY
|
9.0 | IC50 | 2 | — | |
IWPVUHHCWGVPNJ
|
9.0 | IC50 | 5 | Yes | |
JGNYWVKGPUWQDG
|
9.0 | IC50 | 2 | — | |
JVCWPUFNLFSKFS
|
9.0 | IC50 | 5 | — | |
KLHJDCUHOKZNOP
|
9.0 | IC50 | 5 | Yes | |
LBEJYFVJIPQSNX
|
9.0 | IC50 | 4 | — | |
MADCXGNPDBWPLM
|
9.0 | Ki | 25 | — | |
MEBULVBTXSYJKD
|
9.0 | IC50 | 3 | — |