Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JFYAFMMSOVKSEU
|
9.3 | IC50 | 4 | — | |
NKKNQMFHKZEGQU
|
9.3 | IC50 | 5 | — | |
VMAAFUOXTWPYRN
|
9.3 | IC50 | 9 | Yes | |
ZEMQCNHEKKILBX
|
9.3 | IC50 | 3 | — | |
WMWHVTDZNIVNIE
|
9.3 | IC50 | 9 | — | |
ORBLOJJZDLUQDF
|
9.3 | IC50 | 4 | — | |
AYVATFZLZLWIPA
|
9.3 | IC50 | 3 | — | |
BJYQLWPTBHMZKP
|
9.2 | IC50 | 5 | — | |
FJXHHPBKCWCXDJ
|
9.2 | IC50 | 3 | — | |
VDTAJUONJQNBDK
|
9.2 | IC50 | 2 | — | |
QIILXVJHCJSXQI
|
9.2 | IC50 | 3 | — | |
AJFKYSBQAUFOAW
|
9.2 | IC50 | 3 | — | |
FGOGRVVUAJAJDC
|
9.2 | Kd | 2 | — | |
FJWADKUXOQKYQJ
|
9.2 | IC50 | 2 | — | |
GLVVTFVSJIVSIH
|
9.2 | IC50 | 3 | — | |
JOGIYNFTOOGHNQ
|
9.2 | IC50 | 3 | — | |
KPKVXBUKMZIGPN
|
9.2 | IC50 | 3 | — | |
KSJNXKBKMYLRSO
|
9.2 | IC50 | 3 | — | |
OPWIMESOOZSXGC
|
9.2 | IC50 | 2 | — | |
QKFZNOQWHCBRSM
|
9.2 | Kd | 2 | — | |
SRCLLEDPPXOXGH
|
9.2 | IC50 | 3 | — | |
ZRZMENVDJBJBOY
|
9.2 | IC50 | 3 | — | |
WTKYHVUVQSLNBW
|
9.2 | IC50 | 6 | — | |
KZRKENBHNLTBEV
|
9.2 | IC50 | 2 | — | |
QYUAZFYQXCJXEM
|
9.2 | IC50 | 3 | — | |
DUKZDMUZDDNVFF
|
9.2 | IC50 | 3 | — | |
VXLAKHWYGRKCGI
|
9.2 | IC50 | 9 | — | |
FTEUGWHCWRSIJU
|
9.2 | IC50 | 3 | — | |
GVFQHBBRWBJGNU
|
9.2 | IC50 | 5 | — | |
LDRYCDRIKRFDRD
|
9.2 | IC50 | 5 | Yes | |
LIFJGDQDPHYFQJ
|
9.2 | Kd | 2 | — | |
MINWMNHFXQZNMG
|
9.2 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
9.2 | Kd | 220 | — | |
OXRQZPOYHSRCIB
|
9.2 | IC50 | 3 | — | |
QKXDICQFNATVHN
|
9.2 | IC50 | 3 | — | |
RKSPQOPBECGSGM
|
9.2 | IC50 | 3 | — | |
WBVTVMHUUOONFL
|
9.2 | IC50 | 2 | — | |
AJLZQJOCQFFRQL
|
9.1 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
9.1 | IC50 | 49 | Yes | |
YAGLZRLKRDTHPW
|
9.1 | IC50 | 4 | — | |
BGVQPQHIUOTLBT
|
9.1 | Kd | 6 | — | |
JGIUBJWBTUOQHP
|
9.1 | IC50 | 4 | — | |
QZIMFEZMFNJUKH
|
9.1 | IC50 | 4 | — | |
IHLNWRDTNQHABM
|
9.1 | Ki | 3 | — | |
XSLUZOLUJPDNGT
|
9.1 | IC50 | 3 | — | |
CFBKGVOKLIQQJD
|
9.1 | IC50 | 3 | — | |
HOYRWTWZUFFACV
|
9.1 | Ki | 28 | — | |
HXUCFPZSRWJRRN
|
9.1 | IC50 | 3 | — | |
KZVISSXNPKKESH
|
9.1 | IC50 | 3 | — | |
MCOWNEICYXDEPL
|
9.1 | IC50 | 3 | — |