Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BTIIUKSFWMYFNV
|
8.1 | IC50 | 6 | — | |
DTHWSLYDAOOPOE
|
8.1 | IC50 | 4 | — | |
GACBELOLIOXYRT
|
8.1 | IC50 | 4 | Yes | |
JPKSISIJPSXDLA
|
8.1 | IC50 | 10 | Yes | |
KABXDGRHTDMABC
|
8.1 | IC50 | 3 | — | |
MVAYPHGEGDDSJN
|
8.1 | IC50 | 6 | — | |
MZOIOQHNRFBXRZ
|
8.1 | IC50 | 3 | — | |
OEZUXIBNCYTQAV
|
8.1 | IC50 | 5 | Yes | |
QICYOJLQEZXOEU
|
8.1 | IC50 | 3 | — | |
SSMPZXRXMBEUFU
|
8.1 | IC50 | 4 | — | |
ZYBHGENFQHMBLJ
|
8.1 | IC50 | 4 | — | |
ZOHLAZXVTPODGE
|
8.0 | IC50 | 4 | — | |
HGZYVJNUFKTDLR
|
8.0 | IC50 | 2 | — | |
JYBQEMYHVMILOJ
|
8.0 | IC50 | 5 | — | |
LKMNVWCDUCOIDP
|
8.0 | IC50 | 2 | — | |
MMOZHTDOCYODPM
|
8.0 | IC50 | 4 | — | |
CUDRWVZLQYDBKU
|
8.0 | IC50 | 4 | — | |
FXTJCTYAPOCFAC
|
8.0 | IC50 | 4 | — | |
QJNHGKZWLRDZGJ
|
8.0 | IC50 | 2 | — | |
CNWWATUNBGEOQE
|
8.0 | IC50 | 3 | Yes | |
LFJJSPZZCOIAAO
|
8.0 | IC50 | 2 | — | |
QWFWQJOFUNDIAZ
|
8.0 | IC50 | 7 | — | |
SJBXHRBUEGPULP
|
8.0 | IC50 | 4 | — | |
APKGZIMGNRKAIK
|
8.0 | IC50 | 4 | — | |
AYJBHLUSGLQYDG
|
8.0 | Ki | 16 | — | |
BJTVHTAPKJNNGR
|
8.0 | IC50 | 3 | — | |
BRTHUECZMVKNMQ
|
8.0 | Ki | 31 | — | |
CIDVBRKDJFCKQF
|
8.0 | IC50 | 2 | — | |
DJOJKIGNNDWGRS
|
8.0 | Ki | 13 | — | |
DXJBIXWCJZKEHQ
|
8.0 | IC50 | 4 | — | |
FMECAVUOMUCKKM
|
8.0 | IC50 | 3 | Yes | |
GKJQWSMDZOJDIN
|
8.0 | IC50 | 3 | — | |
GQGMUKOYILWOIQ
|
8.0 | Ki | 25 | — | |
GWOSGFTZTVFDGQ
|
8.0 | IC50 | 5 | Yes | |
HGCJKDOLUCMPFE
|
8.0 | IC50 | 5 | — | |
HSYSSKFCQHXOBP
|
8.0 | IC50 | 4 | — | |
JCZBWICLNFNCMR
|
8.0 | Ki | 9 | — | |
KFRUZRAQPBNGME
|
8.0 | IC50 | 3 | Yes | |
LOLPPWBBNUVNQZ
|
8.0 | IC50 | 97 | Yes | |
LPILBMJJRGTKOQ
|
8.0 | Ki | 27 | — | |
MWOBEOJMSDHMFO
|
8.0 | IC50 | 3 | — | |
OQNPAZRZCXFOBC
|
8.0 | Ki | 11 | — | |
OSEYUXXMDLYZKE
|
8.0 | IC50 | 5 | Yes | |
OSIDXFCEXZWGRW
|
8.0 | IC50 | 4 | Yes | |
OTLBXDXENSMYGU
|
8.0 | IC50 | 2 | — | |
OVTHZKRCTBBAOW
|
8.0 | IC50 | 5 | Yes | |
QHWYQHKGOYXAON
|
8.0 | IC50 | 3 | — | |
QOMGQLZYIUPQLG
|
8.0 | IC50 | 7 | — | |
RPUUVOATUZVRNA
|
8.0 | IC50 | 3 | — | |
RRGONMPXYOQEDE
|
8.0 | IC50 | 4 | — |