Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZRKHDIABAALLSW
|
8.1 | IC50 | 3 | — | |
APPUYFNVFFWYFM
|
8.1 | IC50 | 4 | — | |
NEZRLVDPFUFEKB
|
8.1 | IC50 | 4 | — | |
NMQCDRLEHHKROH
|
8.1 | IC50 | 2 | — | |
BHSOPYVVEZFHDB
|
8.1 | IC50 | 25 | Yes | |
DCTBPIBEQFLAOQ
|
8.1 | Ki | 13 | — | |
GBJVVSCPOBPEIT
|
8.1 | Kd | 13 | Yes | |
GTVWQFJFCAUNFY
|
8.1 | IC50 | 2 | — | |
HEUSUIRCBWROMH
|
8.1 | Ki | 64 | — | |
ICVHMFOFVOYFPB
|
8.1 | IC50 | 3 | — | |
KJOZOAQMGSIFNM
|
8.1 | IC50 | 4 | — | |
KXGKWKJLQVNQML
|
8.1 | IC50 | 3 | Yes | |
LGHBDVLAHHANMX
|
8.1 | Ki | 53 | — | |
LRLDYTTWQIFWBD
|
8.1 | Ki | 25 | — | |
MIWWARHIDNFXAZ
|
8.1 | IC50 | 6 | — | |
OEOVBBKVSXNPSX
|
8.1 | IC50 | 3 | — | |
PPPOUAQYRUUFNJ
|
8.1 | IC50 | 4 | — | |
QWIXHSWNLCNTEE
|
8.1 | Ki | 4 | Yes | |
RAPYFGJGASETOS
|
8.1 | Ki | 11 | — | |
SAEGVASGMTZGFI
|
8.1 | IC50 | 2 | — | |
SLKCVFPEQGHNSI
|
8.1 | Ki | 29 | — | |
TULDPDLFHDYJMU
|
8.1 | IC50 | 4 | — | |
TZOUNCJSFSDDCR
|
8.1 | IC50 | 5 | Yes | |
UZYXETLFKQALDE
|
8.1 | IC50 | 3 | — | |
WHDGQRKUPDYCCN
|
8.1 | IC50 | 2 | — | |
WLAVZAAODLTUSW
|
8.1 | IC50 | 7 | — | |
XLFNLJYGUOLEJS
|
8.1 | IC50 | 26 | — | |
ZAARMHXLYCHRAK
|
8.1 | Ki | 20 | — | |
ZOTXBRHWIDKKFO
|
8.1 | IC50 | 4 | Yes | |
ZUNNOMIILKKVTF
|
8.1 | IC50 | 3 | — | |
IKQPJOFHAZFMNC
|
8.1 | IC50 | 4 | — | |
UXYIPHKBTFKDMP
|
8.1 | IC50 | 3 | — | |
WDAHGVLBPINGHW
|
8.1 | IC50 | 6 | — | |
BPFIPYIIVJLOML
|
8.1 | IC50 | 4 | — | |
KEDANNMRCOENMZ
|
8.1 | IC50 | 7 | — | |
KVUCOURZIKDXHZ
|
8.1 | IC50 | 4 | — | |
LYYOHGCLJGVKGA
|
8.1 | IC50 | 2 | — | |
FDCKDXZISZRERO
|
8.1 | IC50 | 5 | — | |
IPOSOQDPXNYXKP
|
8.1 | IC50 | 4 | — | |
JHVBIUJTSAGFKH
|
8.1 | IC50 | 2 | — | |
KYCKKSZMVINEPM
|
8.1 | IC50 | 4 | — | |
MDXPQQJSGHVAGT
|
8.1 | IC50 | 5 | — | |
WDFZKMQYTGAITH
|
8.1 | IC50 | 4 | — | |
XPFFDDFVHAFKNR
|
8.1 | IC50 | 3 | — | |
LBWBNPCQUXPCDH
|
8.1 | IC50 | 4 | — | |
PIELNOLQJZOXMR
|
8.1 | IC50 | 2 | — | |
RAPSXYUJSKOFLB
|
8.1 | IC50 | 4 | — | |
UZISGDYRMAXEPZ
|
8.1 | IC50 | 5 | — | |
AOILZWVIBHVMLR
|
8.1 | IC50 | 4 | — | |
AOLQSKKQHIKRMB
|
8.1 | Ki | 3 | Yes |