Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YVAPXKWBCBCTDS
|
8.2 | IC50 | 4 | — | |
ZXQPAYCROYPEFR
|
8.2 | IC50 | 4 | Yes | |
FVPYEAORCOKOLV
|
8.2 | IC50 | 6 | — | |
MQQJPZHXGJGMDE
|
8.2 | IC50 | 3 | — | |
GMYYMEOGFRKSFS
|
8.2 | Ki | 29 | — | |
HKZKELVPGXJIMW
|
8.2 | Ki | 41 | — | |
JJXRAZVLEQHSOL
|
8.2 | IC50 | 4 | — | |
JRJKATLTRNXYCE
|
8.2 | IC50 | 4 | — | |
KWSZYBNXNYRQCC
|
8.2 | Ki | 21 | — | |
MIOQFVQXGRHCSR
|
8.2 | IC50 | 4 | — | |
MQRDVGBWWVWMEN
|
8.2 | Ki | 47 | — | |
UIARLYUEJFELEN
|
8.2 | IC50 | 2 | — | |
WDARYLSSWBWVCU
|
8.2 | Ki | 49 | — | |
WIXFZICRDRQMNT
|
8.2 | IC50 | 4 | — | |
ZFKQQXLECNVLOF
|
8.2 | IC50 | 7 | — | |
GBLBJPZSROAGMF
|
8.2 | IC50 | 3 | — | |
LFKPJUFFMOTFRX
|
8.2 | IC50 | 6 | — | |
ZXSGJKRDMSVFSU
|
8.2 | IC50 | 3 | — | |
DLPARMNJOHFOLU
|
8.2 | IC50 | 14 | Yes | |
NBIOGGWEVWYBFI
|
8.2 | IC50 | 4 | — | |
QHNQSGOQPWOVDK
|
8.2 | IC50 | 2 | — | |
QQTWEWAFAIDGJB
|
8.2 | IC50 | 4 | — | |
LZOJVTCTBSNNNT
|
8.2 | IC50 | 4 | — | |
BGFQHBDQBASGDN
|
8.2 | IC50 | 4 | — | |
DLFSPMHGSMXBGE
|
8.2 | IC50 | 2 | — | |
MHITTXFPZXWLMH
|
8.2 | Kd | 6 | — | |
BFZLDRFGXXMKES
|
8.2 | IC50 | 5 | Yes | |
BYQDPWAYLMNNKF
|
8.2 | IC50 | 5 | Yes | |
DBDOMJWNBDLGSW
|
8.2 | IC50 | 3 | — | |
FQXJVZZKZWSHEQ
|
8.2 | IC50 | 4 | Yes | |
HQPNLIKXAPLWBQ
|
8.2 | IC50 | 12 | Yes | |
JNROOHWIIJBSJF
|
8.2 | Ki | 2 | Yes | |
JWZRVKDTKFYYDV
|
8.2 | IC50 | 5 | Yes | |
MPVGZUGXCQEXTM
|
8.2 | Kd | 61 | Yes | |
OZLZIPAXURDELS
|
8.2 | IC50 | 3 | — | |
PPXJBXNWKBRGTA
|
8.2 | IC50 | 2 | — | |
SDOPLVMVOKIZQS
|
8.2 | Ki | 2 | — | |
SFNDRKNZETUTKF
|
8.2 | IC50 | 5 | Yes | |
TWYCZJMOEMMCGC
|
8.2 | IC50 | 6 | Yes | |
WQLWLOMHWYQNFN
|
8.2 | IC50 | 4 | — | |
WVVCBUMOFSHDAJ
|
8.2 | IC50 | 3 | — | |
MAQBPYJYNOISMO
|
8.1 | IC50 | 4 | Yes | |
QCKKTDVCCCBGDD
|
8.1 | IC50 | 8 | — | |
QEAUPAREISBURF
|
8.1 | IC50 | 4 | — | |
QGGLESNNYLSYEA
|
8.1 | IC50 | 3 | — | |
YTEDDIJNHJDCLR
|
8.1 | IC50 | 4 | — | |
HGZYVJNUFKTDLR
|
8.1 | IC50 | 2 | — | |
KJVSTAAHJQPRFJ
|
8.1 | IC50 | 3 | — | |
RSRQFBNVFQZQRN
|
8.1 | IC50 | 2 | — | |
TUSFBIZKPNHLKT
|
8.1 | IC50 | 4 | — |