Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RHAMYMXUVZEEJR
|
8.3 | IC50 | 4 | — | |
RHGZQGXELRMGES
|
8.3 | IC50 | 8 | Yes | |
SBLIKFBWCULFJM
|
8.3 | IC50 | 2 | — | |
SECLOTHQGDJSCB
|
8.3 | IC50 | 5 | Yes | |
VWBUFGGJMMUSBL
|
8.3 | IC50 | 4 | — | |
WUWDLXZGHZSWQZ
|
8.3 | Ki | 41 | — | |
XLZFINWQTYEKJR
|
8.3 | IC50 | 5 | Yes | |
XMWHZKQZVIMLTH
|
8.3 | IC50 | 3 | — | |
YBOOAZFLAUPOKA
|
8.3 | Ki | 3 | — | |
YKDDWNDRNJMVDF
|
8.3 | IC50 | 4 | — | |
ZFBBKOBKYNRTOS
|
8.3 | IC50 | 4 | — | |
PXHDQHNAGHIZGO
|
8.3 | IC50 | 4 | — | |
CPNQAVXQGZKRMM
|
8.3 | IC50 | 4 | — | |
CXQHYVUVSFXTMY
|
8.3 | IC50 | 154 | — | |
GTDOWKUTGWWIFA
|
8.3 | IC50 | 3 | — | |
IDQYDZHQPMPCHM
|
8.3 | IC50 | 4 | — | |
LODWOBAYUQRWKD
|
8.3 | IC50 | 7 | — | |
OUSFTKFNBAZUKL
|
8.3 | Kd | 58 | Yes | |
PWOIRDUWFWWFMT
|
8.3 | IC50 | 4 | — | |
QTHCAAFKVUWAFI
|
8.3 | IC50 | 23 | — | |
XYSYRHAUHUPOHK
|
8.3 | IC50 | 4 | — | |
ZYPFDFDWAFKPBY
|
8.3 | IC50 | 3 | — | |
CTNPALGJUAXMMC
|
8.3 | Kd | 151 | — | |
DYDGFQGBJUDGKC
|
8.3 | IC50 | 4 | — | |
FLFGOZHEFLZZRQ
|
8.3 | IC50 | 3 | — | |
GKTJDVXAUIHAML
|
8.3 | IC50 | 4 | — | |
QYCFHBDOJSLVRL
|
8.3 | Kd | 5 | — | |
ROFVRNNNZDBODT
|
8.3 | Kd | 2 | — | |
USMAPSJMQVFIAW
|
8.3 | IC50 | 2 | — | |
YCNFDYPECZUZNM
|
8.3 | IC50 | 4 | — | |
CBJZWQSCZBRXDC
|
8.3 | IC50 | 4 | — | |
GEGOZUGICMLWRA
|
8.3 | IC50 | 3 | — | |
HDRSWNSYJOUCLI
|
8.3 | IC50 | 3 | — | |
AOILZWVIBHVMLR
|
8.2 | IC50 | 4 | — | |
DYMOVSCTFZROSX
|
8.2 | IC50 | 3 | — | |
ZYQKMYRXVHUATB
|
8.2 | Kd | 4 | — | |
UBUCCNWQOAYWFT
|
8.2 | IC50 | 4 | — | |
WTASWEBTFCSOFZ
|
8.2 | IC50 | 2 | — | |
NKTOEINNBIDTOF
|
8.2 | Kd | 2 | — | |
CQMZJAORBQTGTR
|
8.2 | IC50 | 4 | — | |
FIJWNTPHEHDJQG
|
8.2 | IC50 | 6 | Yes | |
IWXVPEORISOBQZ
|
8.2 | IC50 | 3 | — | |
KENMZDPHYLZVEW
|
8.2 | IC50 | 5 | Yes | |
KYEFPHMQFQFRLZ
|
8.2 | IC50 | 3 | — | |
LTGMTZWRANBXGI
|
8.2 | IC50 | 3 | — | |
PQJDGKYKJGBRBM
|
8.2 | Ki | 5 | Yes | |
QWLOMYFDXCOOFH
|
8.2 | IC50 | 5 | Yes | |
SIEQAYSHYKILTK
|
8.2 | IC50 | 3 | — | |
XJXPKTHMXWGQPH
|
8.2 | IC50 | 5 | — | |
YADAQXVHBLKOIU
|
8.2 | IC50 | 4 | — |