Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UQRCJCNVNUFYDX
|
8.4 | Kd | 27 | — | |
WDDLXDTWOAENKE
|
8.4 | IC50 | 5 | Yes | |
HNPGAOXOTQQSMN
|
8.4 | IC50 | 2 | — | |
ZHQZACQNPQRBGO
|
8.4 | IC50 | 4 | — | |
GEDYWUPVBNHAFW
|
8.4 | IC50 | 2 | — | |
JBGGXHXCKFGYPP
|
8.4 | IC50 | 3 | — | |
OVCGZYQGQZKDFH
|
8.4 | IC50 | 2 | — | |
ZVKWOODYBNGMEY
|
8.4 | IC50 | 4 | — | |
WINHZLLDWRZWRT
|
8.4 | IC50 | 201 | Yes | |
MGSYURQJRSJRFB
|
8.4 | Kd | 5 | — | |
PRABTKJJUJZVNX
|
8.4 | IC50 | 4 | — | |
VEVUBFZLKUNGER
|
8.4 | IC50 | 5 | — | |
ZEXUWQNOOJARPB
|
8.4 | IC50 | 2 | — | |
XGWKKUQOFQDOKM
|
8.3 | IC50 | 3 | — | |
AGYRCBTVZCTMOP
|
8.3 | IC50 | 4 | — | |
MJHOMTRKVMKCNE
|
8.3 | IC50 | 12 | — | |
MSSYEZHHVYFPOJ
|
8.3 | IC50 | 2 | — | |
YHELBFBDLFOCAS
|
8.3 | IC50 | 4 | — | |
DHCWIUCAJNMGDF
|
8.3 | IC50 | 4 | — | |
JPMVRYCJGBFRDG
|
8.3 | IC50 | 4 | — | |
CVWXJKQAOSCOAB
|
8.3 | IC50 | 35 | — | |
DVPVWROTHYIYLX
|
8.3 | IC50 | 3 | — | |
PNFHXTSCXQDAOI
|
8.3 | IC50 | 2 | — | |
VWVYILCFSYNJHF
|
8.3 | IC50 | 49 | — | |
YSCRAUWGPPUZRI
|
8.3 | IC50 | 4 | — | |
FXPKSABYJKCHOV
|
8.3 | IC50 | 4 | — | |
LOMPHWBCBDXNOY
|
8.3 | IC50 | 4 | — | |
NEQZWEXWOFPKOT
|
8.3 | IC50 | 9 | Yes | |
ODPGGGTTYSGTGO
|
8.3 | Kd | 153 | — | |
ALKJNCZNEOTEMP
|
8.3 | Kd | 55 | — | |
GALVWTFFXPRMQM
|
8.3 | Ki | 20 | — | |
HWXPNIATGYCXGR
|
8.3 | IC50 | 2 | — | |
HZIZEKOMOILAJT
|
8.3 | IC50 | 6 | Yes | |
ISVHLTLEHRZKJC
|
8.3 | Ki | 19 | — | |
IVZNWJUHDBLKKT
|
8.3 | IC50 | 2 | — | |
IVZNWJUHDBLKKT
|
8.3 | IC50 | 2 | — | |
JLWGOAGEDWMEBT
|
8.3 | IC50 | 10 | — | |
JLWGOAGEDWMEBT
|
8.3 | IC50 | 10 | — | |
JQDTYPFSLIFJAT
|
8.3 | IC50 | 5 | Yes | |
KCCWVRNMXATDGV
|
8.3 | IC50 | 3 | — | |
MKSQDWBNZVGINB
|
8.3 | Ki | 4 | Yes | |
MWUFVYLAWAXDHQ
|
8.3 | IC50 | 2 | — | |
MZHPEELZCYWEHG
|
8.3 | IC50 | 6 | — | |
NAYBZWXBFYYQSG
|
8.3 | IC50 | 3 | — | |
NRGYZNJPCGRCLV
|
8.3 | Ki | 52 | — | |
NRZYTPAJGVTKIM
|
8.3 | Ki | 38 | — | |
OEVGYUXYZSTGNX
|
8.3 | Ki | 2 | Yes | |
OPVYNMNWPXOEJX
|
8.3 | IC50 | 4 | Yes | |
QTTGVGLTCILDCA
|
8.3 | IC50 | 7 | — | |
QZQGXMDLWJNGQH
|
8.3 | IC50 | 4 | — |