Target Details
| UniProt AC | P36888 |
|---|---|
| Gene Symbol | FLT3 |
| Protein Name | Receptor-type tyrosine-protein kinase FLT3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 2,188
- Clinical molecules 305
- Avg pChEMBL 7.53
KEGG Pathways (8)
Associated Diseases (3)
Active Molecules (2,188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WMZGRDMNDXPHMF
|
10.3 | Kd | 2 | — | |
DSWGFGIRFVKDCY
|
10.3 | IC50 | 2 | — | |
CXWKPXGAGKBITA
|
10.0 | IC50 | 3 | — | |
LYHDXABKNJMNEZ
|
10.0 | Ki | 10 | — | |
MBWHJBDHRADERX
|
10.0 | IC50 | 4 | — | |
YGDAYHUWESEYBV
|
9.9 | Kd | 2 | — | |
YIMGMFZUFRVXJG
|
9.9 | IC50 | 2 | — | |
AVMGEAZKDWAZIC
|
9.9 | IC50 | 3 | — | |
GZNUMHPRTTZGTC
|
9.8 | Kd | 3 | — | |
OTAZAWFIQUEVLG
|
9.8 | Kd | 3 | — | |
UUVMNPKFPGJBNX
|
9.8 | Ki | 10 | — | |
FAWULGGSSGGIAH
|
9.8 | IC50 | 2 | — | |
NEQUYNFKQDRNGP
|
9.8 | IC50 | 3 | — | |
IQBCZHKBLZWXEM
|
9.8 | Kd | 3 | — | |
VMZCRJAQNNOYPK
|
9.8 | Kd | 2 | — | |
LAZZFPCNZBTRIQ
|
9.8 | IC50 | 3 | — | |
SNNSTEZDXSIKQW
|
9.7 | Kd | 3 | — | |
JISLYHZGPUPOHU
|
9.7 | Ki | 8 | — | |
VFNJLPYDAYDGKC
|
9.7 | IC50 | 5 | — | |
XBBZAHDOGBGKGM
|
9.7 | IC50 | 5 | Yes | |
NAYMGHBSMQSCDC
|
9.7 | IC50 | 4 | — | |
QSSMDRNGJZDMSQ
|
9.7 | Kd | 3 | — | |
ZQKNIPQNEVNCDY
|
9.6 | Kd | 8 | — | |
IALDYVNFZAPNJV
|
9.5 | Kd | 11 | — | |
GTQSNWXKTIFPBY
|
9.5 | IC50 | 5 | — | |
GYIJQQCWXZLRDA
|
9.5 | IC50 | 2 | — | |
HTJGFHHVVPNDMR
|
9.5 | Kd | 6 | — | |
PBNPHBXRMOAALS
|
9.5 | Kd | 2 | — | |
SINJOIVMLYFADD
|
9.5 | IC50 | 5 | — | |
WEHOMMKULWQPKY
|
9.5 | IC50 | 3 | — | |
FUFJXODRNRQIRI
|
9.5 | Kd | 2 | — | |
JGWMRHPAGIJSBO
|
9.5 | IC50 | 3 | — | |
TWWKXZDIDHDHRF
|
9.4 | IC50 | 7 | — | |
YISMQBFJYDFMAL
|
9.4 | IC50 | 46 | — | |
TZRFJDYUNMZHNZ
|
9.4 | IC50 | 3 | — | |
YEZSPJXJBLNYQO
|
9.4 | Kd | 3 | — | |
UOYOWVPLBRMQFZ
|
9.4 | IC50 | 3 | — | |
BHXZFEQWQQPISU
|
9.4 | Kd | 2 | — | |
FOONBYIHFUMRSX
|
9.4 | Ki | 12 | — | |
HCHLTTBJHNWMPS
|
9.4 | Kd | 2 | — | |
NCPGPVUTWKUPPM
|
9.4 | Kd | 2 | — | |
ULCJFJXVIGNWMX
|
9.4 | Kd | 2 | — | |
YEPNVBNYCRGZRX
|
9.4 | Ki | 26 | — | |
GMAFXYZWTSGYMU
|
9.4 | IC50 | 4 | — | |
NXRKPNCKZKIFMK
|
9.3 | IC50 | 2 | — | |
NPLHHQHEODJUBY
|
9.3 | IC50 | 6 | — | |
MJGKLMMMXSNBCX
|
9.3 | Kd | 3 | — | |
OPWLMVVARKPWEA
|
9.3 | IC50 | 3 | — | |
SXWMIXPJPNCXQQ
|
9.3 | IC50 | 4 | — | |
BDPBZUHWAVABDM
|
9.3 | Ki | 11 | — |