Target Details
| UniProt AC | P36776 |
|---|---|
| Gene Symbol | LONP1 |
| Protein Name | Lon protease homolog, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00004 (AAA) PF05362 (Lon_C) PF22667 (Lon_lid) PF02190 (LON_substr_bdg) |
Summary
- Multi-target molecules 8
- Clinical molecules 0
- Avg pChEMBL 7.03
Associated Diseases (1)
Active Molecules (8)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XQCVLFKVFQVTPX
|
7.7 | IC50 | 20 | — | |
ZTZIILNFYPSLFR
|
7.5 | IC50 | 20 | — | |
MWKSRKSEWLRPBL
|
7.2 | Kd | 1075 | — | |
UKWSBIBETQJWIR
|
7.0 | IC50 | 20 | — | |
ILENEQWIGPQYCQ
|
7.0 | IC50 | 20 | — | |
JNOIFOLTDCGUJG
|
6.9 | IC50 | 20 | — | |
GXJABQQUPOEUTA
|
6.7 | IC50 | 47 | — | |
ZCCPLJOKGAACRT
|
6.2 | Kd | 599 | — |