Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BSBQPLUISHJULY
|
8.5 | IC50 | 11 | — | |
CARLZFLTQJQGIP
|
8.5 | IC50 | 3 | — | |
CNIWCJQSFDYIDI
|
8.5 | IC50 | 3 | — | |
CVUXIABNRCIXRF
|
8.5 | IC50 | 2 | Yes | |
CXDZGSNFZYGQSZ
|
8.5 | IC50 | 4 | Yes | |
DLGIXSWHFYBLQG
|
8.5 | IC50 | 2 | — | |
DZSUJUOJJJCWGG
|
8.5 | IC50 | 55 | Yes | |
FGZIONRFHVNRJB
|
8.5 | IC50 | 3 | — | |
FIWBNUYYYKCFHG
|
8.5 | IC50 | 4 | — | |
FPQYONGXMYWJCL
|
8.5 | IC50 | 2 | — | |
FQYLJBVSYHZWLT
|
8.5 | IC50 | 35 | Yes | |
GTHUEDBAWKTNDV
|
8.5 | IC50 | 3 | — | |
HEBQIUUCKUBQCJ
|
8.5 | IC50 | 2 | — | |
HJFDTNBKNJFDQP
|
8.5 | IC50 | 3 | — | |
IOYGAWXBNPFOKF
|
8.5 | IC50 | 3 | — | |
IRVGRHMDHCZIOZ
|
8.5 | IC50 | 4 | — | |
KBUOUGKAAPDJRZ
|
8.5 | IC50 | 2 | — | |
KPVSGWFUYLJRIW
|
8.5 | IC50 | 2 | — | |
LMFNJXLDISVWLF
|
8.5 | IC50 | 5 | — | |
NOLVXPFFXLMLIM
|
8.5 | IC50 | 2 | — | |
OWBPDWHZXAEGMJ
|
8.5 | IC50 | 2 | — | |
PDXLFGGSCODVJA
|
8.5 | Kd | 3 | — | |
PVZJLPGZMRIHCQ
|
8.5 | IC50 | 3 | — | |
RAHBGWKEPAQNFF
|
8.5 | IC50 | 26 | — | |
RAMCMRRBGWIDLK
|
8.5 | IC50 | 8 | Yes | |
SDLZNEBGHGGFNW
|
8.5 | IC50 | 3 | — | |
UDLYZSYBPOFSSA
|
8.5 | IC50 | 2 | — | |
UFSGCADQVRKELP
|
8.5 | IC50 | 3 | — | |
WIICWOVXHJZGNO
|
8.5 | IC50 | 2 | — | |
WQTDKOSNNMUDQK
|
8.5 | IC50 | 5 | — | |
WZZOTDRFRPWXSI
|
8.5 | IC50 | 2 | — | |
XHORJSJFHVABEA
|
8.5 | IC50 | 5 | — | |
XHXOJKOXEKXDSQ
|
8.5 | IC50 | 5 | Yes | |
ZCCJKVBTHCOISJ
|
8.5 | IC50 | 46 | — | |
ZKKRNZFCHLYOFH
|
8.5 | IC50 | 2 | — | |
ZMZOKLZTXMCMNW
|
8.5 | IC50 | 4 | — | |
ZVIWALRWYYSHSU
|
8.5 | IC50 | 3 | — | |
KYABXXGGLXXKNT
|
8.5 | IC50 | 2 | — | |
GKEYKDOLBLYGRB
|
8.5 | IC50 | 3 | — | |
HKZKELVPGXJIMW
|
8.5 | Ki | 41 | — | |
IPIQDJVAZDCFFX
|
8.5 | IC50 | 2 | — | |
LFRLYJOQYBDOIR
|
8.5 | IC50 | 2 | — | |
MCCCQFAOMZMZKE
|
8.5 | IC50 | 52 | — | |
NSKFXNDKPCVDIN
|
8.5 | Ki | 12 | — | |
NVQDLTVJFMBRNP
|
8.5 | IC50 | 2 | — | |
SJMFZIGFOIPNPE
|
8.5 | Ki | 10 | — | |
UUVMNPKFPGJBNX
|
8.5 | IC50 | 10 | — | |
WJWZBQQEQNLYFQ
|
8.5 | Ki | 3 | — | |
WYMDWWZXERLYKQ
|
8.5 | IC50 | 3 | — | |
ALKQTTOWJRBJBP
|
8.5 | IC50 | 2 | — |