Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FARNSAZMRIPYES
|
8.6 | IC50 | 2 | — | |
SANPFBFWRPCKIY
|
8.6 | IC50 | 3 | — | |
SDGGLMMHOSCYCM
|
8.6 | IC50 | 2 | — | |
YTFYNVSEHUSYCW
|
8.6 | IC50 | 4 | — | |
BLNFXBVDIFFNQY
|
8.6 | IC50 | 2 | — | |
BXMUFQGDIWSQBJ
|
8.6 | Ki | 7 | — | |
MGWSCJCLMDQNGB
|
8.6 | IC50 | 2 | — | |
PETGNDYNMCNUKJ
|
8.6 | IC50 | 3 | — | |
PSQQJYVAJZSKPM
|
8.6 | IC50 | 2 | — | |
ROHJEIACUNTGFP
|
8.6 | IC50 | 16 | — | |
STSJLCHGAYUSER
|
8.6 | IC50 | 2 | — | |
VZRIBSCWFNIDIU
|
8.6 | IC50 | 3 | — | |
ZJIOFIWKIMJTMZ
|
8.6 | IC50 | 2 | — | |
BUZZYBLUNDCBEB
|
8.6 | IC50 | 2 | — | |
HZHDGZNDKAIYRX
|
8.6 | IC50 | 2 | — | |
PMCATQTXBPQRSD
|
8.6 | IC50 | 3 | — | |
DNBSBOYLZWOFKX
|
8.6 | IC50 | 2 | — | |
HNAKAPUKEWMJOX
|
8.6 | IC50 | 2 | — | |
HZMLMSFEXUJVAY
|
8.6 | IC50 | 2 | Yes | |
JNLSTLQFDDAULK
|
8.6 | IC50 | 4 | — | |
NMGSBNKYPAIWOG
|
8.6 | IC50 | 3 | — | |
OLGSVSPNJXGSAD
|
8.6 | IC50 | 5 | Yes | |
PMNKHDAXQLPDIQ
|
8.6 | IC50 | 2 | — | |
SXGZAYZKUGJQPT
|
8.6 | IC50 | 2 | — | |
TTXOTMLADFPMGH
|
8.6 | IC50 | 2 | — | |
VXXXFNQITZZUER
|
8.6 | IC50 | 2 | — | |
YRQFTXBTINKLCO
|
8.6 | IC50 | 2 | — | |
UVZNMKLHIOHOBN
|
8.6 | IC50 | 3 | — | |
MDPMAXSABUPRJI
|
8.6 | IC50 | 2 | — | |
MQCFWAKOIXTUQK
|
8.6 | IC50 | 2 | Yes | |
PKCCJOWYVJUGKD
|
8.6 | IC50 | 3 | — | |
QATOHKJFHXOHIB
|
8.6 | IC50 | 2 | Yes | |
XHPCNYYPHRXXOG
|
8.6 | IC50 | 2 | — | |
CICHSTJOLCRZKB
|
8.5 | Kd | 2 | — | |
GHHLGOSWKKKPAV
|
8.5 | IC50 | 2 | — | |
IDBPJJQGJZOVMW
|
8.5 | IC50 | 2 | Yes | |
JLBAXNKYJZOYGQ
|
8.5 | IC50 | 4 | Yes | |
MLLQJNIKDWEEFT
|
8.5 | IC50 | 6 | — | |
NMJILYFXNANMKC
|
8.5 | IC50 | 3 | — | |
NQWHKZFLRJPUMS
|
8.5 | IC50 | 4 | — | |
SOBMUPLZQRAPEL
|
8.5 | IC50 | 2 | — | |
XIQQPHOWVZOQQP
|
8.5 | IC50 | 4 | — | |
CPTVWYCNJGYSDW
|
8.5 | IC50 | 3 | — | |
MAWWXEIKARIPSX
|
8.5 | IC50 | 2 | — | |
VUKUZGSFRAYWPM
|
8.5 | IC50 | 2 | — | |
AMHUBFWCCMLLCJ
|
8.5 | IC50 | 15 | — | |
APMQKHHNTLVDQD
|
8.5 | IC50 | 6 | Yes | |
AWXSQBQLENVFPN
|
8.5 | IC50 | 2 | — | |
BGHOGQNFMBHPKJ
|
8.5 | IC50 | 2 | Yes | |
BMFHAIYLTOVZTR
|
8.5 | IC50 | 2 | — |