Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KRIMNORKYPAQGO
|
8.7 | IC50 | 2 | — | |
MJMJYGWCNKSGSI
|
8.7 | IC50 | 2 | — | |
MYMJRZXUXNYPIX
|
8.7 | IC50 | 2 | — | |
NPUAKRMYWJOTLS
|
8.7 | IC50 | 2 | — | |
OASNOJDJXITQNB
|
8.7 | IC50 | 2 | — | |
OHHGYJBFPVJURR
|
8.7 | IC50 | 2 | — | |
PHUIVAKJVUJLDO
|
8.7 | IC50 | 3 | — | |
QCARBCGPQHFPOS
|
8.7 | IC50 | 2 | — | |
SNRUTMWCDZHKKM
|
8.7 | IC50 | 4 | — | |
VOZWUTXGVBZOLP
|
8.7 | IC50 | 2 | Yes | |
VRKCCBOVUKMTIE
|
8.7 | IC50 | 4 | — | |
WPHKIQPVPYJNAX
|
8.7 | IC50 | 81 | — | |
WSBZFFNSBMBYQA
|
8.7 | IC50 | 9 | — | |
YEIASMOUYNOXGA
|
8.7 | IC50 | 5 | — | |
ZGDSBEUMPIMXBM
|
8.7 | IC50 | 42 | — | |
CLOKCIDZTVIDMJ
|
8.7 | IC50 | 2 | Yes | |
JPJAUHSLJCUGAH
|
8.7 | IC50 | 4 | — | |
LYHXSDWIWVVZPB
|
8.7 | IC50 | 6 | Yes | |
QDQFGRCUJGQRLD
|
8.7 | IC50 | 3 | — | |
BYYYCNUDMZSOGS
|
8.7 | IC50 | 5 | Yes | |
SIFWORLXBPDHFA
|
8.7 | IC50 | 2 | — | |
AQSSMEORRLJZLU
|
8.7 | IC50 | 34 | Yes | |
JEZNQOLZSHORKU
|
8.7 | IC50 | 2 | — | |
MDNAJFVDTSUEGN
|
8.7 | IC50 | 3 | — | |
SVEZALKOLCCBNB
|
8.7 | IC50 | 2 | — | |
UGEJLCNSVIVALC
|
8.7 | IC50 | 41 | — | |
ZOTWWNJHIZTSQU
|
8.7 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
8.6 | Kd | 151 | — | |
OMPVQOOIKZDYGO
|
8.6 | IC50 | 2 | — | |
QFHBSJJMTUPRMF
|
8.6 | IC50 | 2 | — | |
QQGKEHCROAPVMW
|
8.6 | IC50 | 3 | — | |
SUXYGJZMCWKJJI
|
8.6 | IC50 | 26 | Yes | |
YZBMZVFTUOENSZ
|
8.6 | IC50 | 2 | Yes | |
BCVBGCRLWBQIAF
|
8.6 | IC50 | 2 | — | |
VPXYJYVAKTVLLA
|
8.6 | IC50 | 2 | — | |
DBXOMQJZSQLQED
|
8.6 | IC50 | 12 | — | |
IWBVZILESKBVJL
|
8.6 | IC50 | 6 | — | |
IXIJKXSIADDKHR
|
8.6 | IC50 | 12 | — | |
SPMVMDHWKHCIDT
|
8.6 | IC50 | 30 | — | |
SPMVMDHWKHCIDT
|
8.6 | IC50 | 5 | — | |
WRXMYALXQGBBNT
|
8.6 | IC50 | 2 | — | |
XROVNERVLRWCAV
|
8.6 | IC50 | 3 | — | |
IWBIEKJAAQYGMI
|
8.6 | IC50 | 3 | — | |
SXGZAYZKUGJQPT
|
8.6 | IC50 | 2 | — | |
WEWNFYSPKIFAFJ
|
8.6 | IC50 | 2 | — | |
XDMQGCSGNALEEM
|
8.6 | IC50 | 2 | — | |
ZTLIJXDSHRPKGC
|
8.6 | IC50 | 2 | — | |
ARYDDRNBUXLRQZ
|
8.6 | IC50 | 3 | — | |
AUNHGNQTPLHIRO
|
8.6 | IC50 | 2 | — | |
CRNIURWEBLRATC
|
8.6 | IC50 | 5 | — |