Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HZIZEKOMOILAJT
|
8.8 | IC50 | 6 | Yes | |
CBPRXMDBGJCNJA
|
8.8 | IC50 | 2 | — | |
BYSPSKYBWHPEJW
|
8.8 | IC50 | 6 | — | |
DELFTXSEBVUJAK
|
8.8 | IC50 | 3 | — | |
FOFCTFMFMUVWOA
|
8.8 | IC50 | 3 | — | |
SZSDKEQZCBOVMW
|
8.8 | IC50 | 3 | — | |
UJKFLFOBPZHDJN
|
8.8 | IC50 | 3 | — | |
WYSIIHBXZUVHPY
|
8.8 | IC50 | 2 | Yes | |
BYDMGYUSZLFTLB
|
8.8 | IC50 | 2 | — | |
GJWFUGSRILNJBR
|
8.8 | IC50 | 4 | — | |
KSXXLYFDRDYXJK
|
8.8 | IC50 | 3 | — | |
RGAHTFBLOZYPNE
|
8.8 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
8.8 | IC50 | 8 | — | |
WYLBYVHRCHPXRQ
|
8.8 | IC50 | 3 | — | |
ZQQVWTACALNOAJ
|
8.8 | Ki | 11 | — | |
WCDLCPLAAKUJNY
|
8.8 | IC50 | 8 | — | |
FOKQTIHUENEYBC
|
8.8 | IC50 | 2 | — | |
MRYVITFPRDXAHG
|
8.8 | IC50 | 2 | — | |
NCLNWRLLRGLRTQ
|
8.8 | IC50 | 3 | — | |
PHXJVRSECIGDHY
|
8.8 | IC50 | 59 | — | |
VAWLAPYBUJTXRS
|
8.8 | IC50 | 6 | Yes | |
FLYHUTANLWWHSP
|
8.8 | IC50 | 2 | — | |
SXGZAYZKUGJQPT
|
8.8 | IC50 | 2 | — | |
FCLMAXRVUCVWGI
|
8.8 | IC50 | 2 | — | |
VZQHANSAAHZYGF
|
8.8 | IC50 | 2 | — | |
BRTHUECZMVKNMQ
|
8.7 | IC50 | 7 | — | |
CYVPXDNOIYCAAV
|
8.7 | IC50 | 2 | — | |
KHKKHXIFTCUDNT
|
8.7 | IC50 | 2 | — | |
UHQHOJQDEGMFKV
|
8.7 | IC50 | 2 | — | |
VTBJZDMBUWEQBI
|
8.7 | IC50 | 2 | — | |
WUEVFQBRVSPKLA
|
8.7 | IC50 | 2 | — | |
WYCNEMUMQDPFHP
|
8.7 | IC50 | 2 | — | |
LFKQSJNCVRGFCC
|
8.7 | IC50 | 6 | — | |
MIIRGIJHJBFFEA
|
8.7 | IC50 | 3 | — | |
SIFWORLXBPDHFA
|
8.7 | IC50 | 2 | — | |
SOXNNGFGYDFPDL
|
8.7 | IC50 | 3 | — | |
BWWSAKOFIQJSSK
|
8.7 | IC50 | 4 | — | |
CKRJSIFFXMHDSE
|
8.7 | IC50 | 3 | Yes | |
DOUJIQCJKZYPBP
|
8.7 | IC50 | 3 | — | |
GITNDHUJOBXSCE
|
8.7 | IC50 | 4 | — | |
GBFDLYAUGOZCIP
|
8.7 | IC50 | 2 | — | |
JKDOLJKPWNOURO
|
8.7 | IC50 | 3 | — | |
PLBNUXRJFUCRRW
|
8.7 | IC50 | 2 | — | |
ASUVAFYTTOHJIF
|
8.7 | IC50 | 2 | — | |
BDPBZUHWAVABDM
|
8.7 | IC50 | 11 | — | |
BQNQMLPWBQGGJJ
|
8.7 | IC50 | 2 | — | |
FCPPQNZGDIZFLT
|
8.7 | IC50 | 3 | Yes | |
GZMFYPWWSXGVTC
|
8.7 | Ki | 2 | — | |
HSKISFLIRPOYCF
|
8.7 | IC50 | 5 | — | |
HTMVIKSMELCDMN
|
8.7 | IC50 | 2 | — |