Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GWQQUSRBNJRKLG
|
9.0 | IC50 | 3 | — | |
HJSPWWLBAHRSAY
|
9.0 | IC50 | 2 | — | |
IREATOXCIIIDEG
|
9.0 | Ki | 4 | — | |
IVQYCPCHHYNLKB
|
9.0 | IC50 | 3 | — | |
LYHDXABKNJMNEZ
|
9.0 | IC50 | 10 | — | |
MJJXPCMDOLZDMW
|
9.0 | IC50 | 2 | — | |
MZWXPLVBKPHKNC
|
9.0 | IC50 | 2 | Yes | |
NZUGNTZEMQTKDH
|
9.0 | IC50 | 2 | — | |
UYWCBKUMESQOKL
|
9.0 | IC50 | 5 | — | |
WSHIGLALBLRQGR
|
9.0 | IC50 | 2 | — | |
XYJONLOLMGUYBZ
|
9.0 | IC50 | 6 | — | |
ZAJKUNDNLWGYKD
|
8.9 | IC50 | 3 | — | |
VZRLBUJXKJBRFA
|
8.9 | IC50 | 3 | — | |
FGDPUUPSGZJLCV
|
8.9 | IC50 | 2 | — | |
HPIULPPERVHOJE
|
8.9 | IC50 | 2 | — | |
AISWQGLURAAAKE
|
8.9 | IC50 | 7 | — | |
GUUYUIDTJAWAHO
|
8.9 | IC50 | 4 | — | |
GYWJHWLJQBKSEF
|
8.9 | IC50 | 2 | — | |
NHMWKPIXGXPWGN
|
8.9 | IC50 | 2 | — | |
NZDHEVOTZDNDBN
|
8.9 | IC50 | 2 | — | |
TZSBMAHRPWFGJQ
|
8.9 | IC50 | 2 | — | |
ISVKXCPIKLZVQW
|
8.9 | IC50 | 3 | Yes | |
LMCLMMAYWZRBRH
|
8.9 | IC50 | 2 | — | |
BRTHUECZMVKNMQ
|
8.9 | Ki | 31 | — | |
GJKVMXDBPDDFHI
|
8.9 | Ki | 27 | — | |
GONLMECPQWNPOT
|
8.9 | IC50 | 2 | — | |
KYABXXGGLXXKNT
|
8.9 | IC50 | 2 | — | |
RPDVCUCXMGWTFA
|
8.9 | Ki | 10 | — | |
RTYJMUXLFRYRBU
|
8.9 | Ki | 35 | — | |
VCFDMLBPASGZTP
|
8.9 | Ki | 38 | — | |
BEIAIBOGYLFZCK
|
8.9 | IC50 | 4 | — | |
BEVPJXUTHBNTLS
|
8.9 | IC50 | 3 | Yes | |
DQHFKDYMNMRFQA
|
8.9 | IC50 | 2 | Yes | |
HSAQBRJGYZIVJP
|
8.9 | IC50 | 5 | Yes | |
JRGLHUFNZUQJNB
|
8.9 | IC50 | 2 | — | |
KIVHIZZKZIPROE
|
8.9 | IC50 | 2 | — | |
VKRRGKOVGYHCBL
|
8.9 | IC50 | 2 | — | |
YHYJQEMFCWJMSJ
|
8.9 | IC50 | 2 | Yes | |
YIXJIOOQSSSYGU
|
8.9 | IC50 | 4 | — | |
ZSWBFDGBEZTJRY
|
8.9 | IC50 | 4 | — | |
ZYYNXHSAMWEIKK
|
8.9 | IC50 | 4 | Yes | |
JRHZSLDMBCJCRQ
|
8.9 | IC50 | 2 | — | |
FGPIVIJULBNRBX
|
8.9 | IC50 | 4 | — | |
LIMHWCZODBAXBC
|
8.9 | IC50 | 3 | — | |
DEMGLABBZSLUOH
|
8.8 | IC50 | 3 | — | |
FEWAGHIBDBSVCS
|
8.8 | IC50 | 2 | — | |
IFFBOVLYGJAFKB
|
8.8 | IC50 | 5 | — | |
JBKRHKORBCTVLD
|
8.8 | IC50 | 2 | — | |
QPUJGBSZMTZOCB
|
8.8 | IC50 | 2 | — | |
BHBBGXQSTGBYSZ
|
8.8 | IC50 | 2 | — |