Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XBNLLMKPDMJSKX
|
9.1 | IC50 | 2 | — | |
CTUNMKNUSCLTQS
|
9.0 | IC50 | 2 | — | |
VLTUYLMKVNYVHY
|
9.0 | IC50 | 2 | — | |
VYMBMEPSKRYKBW
|
9.0 | Ki | 2 | — | |
WBFPMZZURZSNBB
|
9.0 | IC50 | 2 | — | |
ZDMGPVTVMCERRZ
|
9.0 | IC50 | 3 | — | |
ZMLDVKWBDWLLML
|
9.0 | IC50 | 2 | — | |
DZFZXPPHBWCXPQ
|
9.0 | IC50 | 12 | — | |
GAKOWURXFQKQGU
|
9.0 | IC50 | 2 | — | |
HWSPZCPLTSAAED
|
9.0 | IC50 | 2 | — | |
JEZNQOLZSHORKU
|
9.0 | IC50 | 2 | — | |
JNEHFOFHMXRLFR
|
9.0 | Ki | 2 | — | |
LZQMVZQCOPEYQN
|
9.0 | IC50 | 2 | — | |
DSYCVJBNOBWEDH
|
9.0 | IC50 | 2 | — | |
VUPUUXMMYXRPFF
|
9.0 | IC50 | 2 | — | |
YOZUNJXPGMAPQP
|
9.0 | IC50 | 2 | — | |
ABXJJVJJEAFTLI
|
9.0 | IC50 | 4 | — | |
AJCUOYPNGRYALV
|
9.0 | IC50 | 2 | — | |
BIGLUOGTKFYENL
|
9.0 | IC50 | 2 | Yes | |
CPZZPVRAQQJBTN
|
9.0 | IC50 | 2 | Yes | |
CREAAGUFOMLCKF
|
9.0 | IC50 | 3 | Yes | |
DHILENNEVBDEMU
|
9.0 | IC50 | 2 | — | |
DJNWXYTWORPJNI
|
9.0 | IC50 | 4 | Yes | |
DVRSTRMZTAPMKO
|
9.0 | IC50 | 10 | Yes | |
DYBGLIINTRJUKT
|
9.0 | IC50 | 2 | — | |
JFGLOXKNWPNMQT
|
9.0 | IC50 | 5 | Yes | |
LXBUSRPKZONHPE
|
9.0 | IC50 | 4 | Yes | |
MQRYORPEARKGSY
|
9.0 | IC50 | 4 | Yes | |
MWDKQVZICDCEDA
|
9.0 | IC50 | 3 | — | |
NECQZMQPXFYVOY
|
9.0 | Ki | 26 | — | |
NKKSIIYIDSJFSX
|
9.0 | IC50 | 3 | Yes | |
OQKMFDJSKWESCR
|
9.0 | IC50 | 4 | Yes | |
ORRHVRJUSPCILV
|
9.0 | Ki | 16 | — | |
PPTQWMQTXBVAHT
|
9.0 | IC50 | 2 | — | |
QYQLAHVYGBJXDH
|
9.0 | IC50 | 2 | — | |
UTVABCSMEKUFLJ
|
9.0 | IC50 | 7 | Yes | |
UXQLMVSZSYZFID
|
9.0 | Ki | 12 | — | |
VCBGNDQGKNIBBK
|
9.0 | IC50 | 6 | Yes | |
WPEWQEMJFLWMLV
|
9.0 | IC50 | 2 | — | |
XBINIPRQWSOQIE
|
9.0 | IC50 | 4 | Yes | |
XXJWYDDUDKYVKI
|
9.0 | IC50 | 52 | — | |
YFIFSHPCXQZADK
|
9.0 | IC50 | 2 | — | |
YJFKREHADGLMHG
|
9.0 | IC50 | 2 | — | |
ZKVQZKJTCLSERL
|
9.0 | IC50 | 2 | Yes | |
ZOKZHFIBKOVHBQ
|
9.0 | IC50 | 2 | — | |
GCUZSJPHOPKZNQ
|
9.0 | IC50 | 2 | — | |
RJOOYQPEJJZEIP
|
9.0 | IC50 | 2 | — | |
RHZNEYIWEJCIRC
|
9.0 | IC50 | 2 | — | |
XLBQFFPUVVTFGK
|
9.0 | IC50 | 3 | — | |
FEMXGYPLUJMECJ
|
9.0 | IC50 | 2 | — |