Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RXZNKADVZBVZKL
|
9.2 | IC50 | 2 | — | |
ZFFOQWCQWWHTIS
|
9.2 | IC50 | 3 | — | |
IFAAYTNDJIPJBZ
|
9.2 | IC50 | 2 | — | |
JYRPSPNQBJTHFR
|
9.2 | IC50 | 2 | — | |
SWGYDVUEALYJJW
|
9.2 | IC50 | 2 | — | |
AQGHUQFARNGYDN
|
9.2 | IC50 | 2 | — | |
CQGCMAIBZGXOAJ
|
9.2 | IC50 | 3 | — | |
FOONBYIHFUMRSX
|
9.2 | IC50 | 12 | — | |
FZUIMQXCCXUHPW
|
9.2 | IC50 | 2 | — | |
IGXWHXJCDUCSBX
|
9.2 | IC50 | 2 | — | |
JBIRTAVBFDUZQN
|
9.2 | IC50 | 2 | — | |
OPTZTHAQEZWUIM
|
9.2 | IC50 | 2 | — | |
WEDWUMJCHQDOEH
|
9.2 | IC50 | 3 | — | |
ZFHLKLQIDSNDHN
|
9.2 | IC50 | 3 | — | |
SSHPGUNPHGPTSE
|
9.1 | IC50 | 2 | — | |
DTHSJRSUDUUQFI
|
9.1 | IC50 | 3 | — | |
CTUNMKNUSCLTQS
|
9.1 | IC50 | 2 | — | |
MEBWIBLSBZGQSC
|
9.1 | IC50 | 3 | — | |
QIZGCINCAAEMBX
|
9.1 | IC50 | 2 | — | |
PAQLCNBPWYBOJT
|
9.1 | IC50 | 5 | — | |
RXVARTZYPOQZBI
|
9.1 | IC50 | 2 | — | |
UAOGCFLMMYQHFB
|
9.1 | IC50 | 2 | — | |
XCTJBNLLBRCFCQ
|
9.1 | IC50 | 2 | — | |
XTZUWEGTTUIMBG
|
9.1 | Ki | 9 | — | |
IMFSTVJNACYASP
|
9.1 | IC50 | 2 | — | |
REYMYGJJLFMJCU
|
9.1 | IC50 | 2 | — | |
RKLGMDOZEOTQEM
|
9.1 | Ki | 12 | — | |
UMBIRSZUCJNBHB
|
9.1 | IC50 | 18 | — | |
WJIAKJKQRZFXIW
|
9.1 | IC50 | 2 | — | |
FIGALARIXLDOBI
|
9.1 | IC50 | 2 | — | |
GCVSOKZESRXLDF
|
9.1 | IC50 | 2 | — | |
GMNBLWOJWJDQBB
|
9.1 | IC50 | 2 | — | |
OHRPYVMGIKIEMB
|
9.1 | IC50 | 2 | — | |
SAUWKRYRSAXLGI
|
9.1 | Ki | 2 | — | |
VZDAKDOJJGVGBR
|
9.1 | IC50 | 2 | — | |
NNYCTPRWKDDLFA
|
9.1 | IC50 | 2 | — | |
XMFJUJPBMXFKQN
|
9.1 | IC50 | 2 | — | |
HQSVYZWDHYEPBY
|
9.1 | IC50 | 2 | — | |
LZICBLBTUMGIRS
|
9.1 | Ki | 2 | — | |
MBRAIJANXVZJAV
|
9.1 | IC50 | 2 | — | |
RZJRJEDTYIELCA
|
9.1 | IC50 | 2 | — | |
SSHPGUNPHGPTSE
|
9.1 | IC50 | 2 | — | |
UMFBYZXXIZIFTP
|
9.1 | IC50 | 2 | — | |
VTZUUFAMKLHHRM
|
9.1 | IC50 | 2 | — | |
AGUVNAJQOHNWNU
|
9.1 | IC50 | 2 | — | |
FNVQWFPDIYQCSF
|
9.1 | IC50 | 8 | Yes | |
GDAJJNYCUJYRBK
|
9.1 | Ki | 2 | — | |
LDYBJNSNFYSDIW
|
9.1 | IC50 | 4 | Yes | |
REWMPRKUAPYNBX
|
9.1 | IC50 | 2 | — | |
WFJQCQNBWDAYSK
|
9.1 | IC50 | 4 | — |