Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SWQMXRJDVZRZBE
|
9.4 | IC50 | 2 | — | |
QGTNBHVHNFUNSQ
|
9.3 | IC50 | 2 | — | |
VCDOUBNPUAACRA
|
9.3 | IC50 | 2 | Yes | |
BIYLXMSIYSWZMT
|
9.3 | IC50 | 4 | — | |
PPUIQOGYMIRZOS
|
9.3 | IC50 | 2 | — | |
LCFJBBWUVXKZGB
|
9.3 | IC50 | 2 | — | |
WUBFAXNVDMCVIO
|
9.3 | IC50 | 12 | Yes | |
NEQZWEXWOFPKOT
|
9.3 | IC50 | 9 | Yes | |
ARFSBNIXMVQEPO
|
9.3 | IC50 | 2 | — | |
CEIYRBYXRSULDG
|
9.3 | IC50 | 4 | Yes | |
COYNQUUUEZTJFP
|
9.3 | IC50 | 2 | — | |
DVHSIXNBKKXFCJ
|
9.3 | IC50 | 2 | — | |
HAWQJVUHZAYNCF
|
9.3 | IC50 | 5 | — | |
KOFXELGVKHKUJR
|
9.3 | IC50 | 3 | — | |
RNHWXYKRVZUXGO
|
9.3 | IC50 | 4 | Yes | |
SFUSDJRVEVLCSW
|
9.3 | IC50 | 2 | — | |
VDTIARDTOLLQLW
|
9.3 | IC50 | 2 | — | |
VMAAFUOXTWPYRN
|
9.3 | IC50 | 9 | Yes | |
AMRDEKYBJXNLRC
|
9.3 | IC50 | 3 | — | |
PIBOSMWVYTUUIX
|
9.3 | IC50 | 3 | — | |
WEMHHXYZAJVSME
|
9.3 | IC50 | 3 | — | |
LFXRUSJBXAQXCD
|
9.3 | IC50 | 2 | — | |
USFUHWQRVTVWKY
|
9.3 | IC50 | 2 | — | |
ZNKAHOBYOWIVNF
|
9.3 | IC50 | 2 | — | |
FZXFZHFLUJFRGT
|
9.3 | IC50 | 2 | — | |
NMMQJLYMIJYIAK
|
9.3 | IC50 | 3 | — | |
WFLJBHIMLGVBCP
|
9.3 | IC50 | 2 | — | |
FYFHKYILOCTNFL
|
9.2 | IC50 | 2 | — | |
IKZHBZBLVAJZJP
|
9.2 | IC50 | 2 | — | |
JQWRPCZUMWGJSB
|
9.2 | IC50 | 2 | — | |
PAHBMDHIMGYJEW
|
9.2 | IC50 | 2 | — | |
VZHPNWDSQYCLOK
|
9.2 | IC50 | 3 | — | |
HJRLGIHYFRRZGA
|
9.2 | IC50 | 2 | — | |
XWFXAJNJXGILIN
|
9.2 | IC50 | 3 | — | |
HSCPAFQDYZFJML
|
9.2 | IC50 | 2 | — | |
NNFDRCGXLJTASH
|
9.2 | IC50 | 4 | — | |
OSZVHJYNXBUVAH
|
9.2 | IC50 | 12 | — | |
PKFMTQRFZPFQOL
|
9.2 | IC50 | 4 | Yes | |
QIZGCINCAAEMBX
|
9.2 | IC50 | 2 | — | |
UKVWGCUKJNZWPI
|
9.2 | Ki | 2 | — | |
ZATGFXTWDKIEKC
|
9.2 | IC50 | 8 | Yes | |
IJIGYLWUTHHVOT
|
9.2 | IC50 | 2 | — | |
KROLCVQARUUHNV
|
9.2 | Ki | 12 | — | |
KUNZDWIFPOMUOX
|
9.2 | Ki | 36 | — | |
NWMPVMMGSHXANZ
|
9.2 | Ki | 58 | — | |
CTUNMKNUSCLTQS
|
9.2 | IC50 | 2 | — | |
QEXZHTIPIXJKTN
|
9.2 | IC50 | 3 | — | |
FGBWIPBEKQBXCP
|
9.2 | IC50 | 2 | — | |
LOCGWCWPUSRMSW
|
9.2 | IC50 | 2 | — | |
LUQXZVFBJJZMSL
|
9.2 | IC50 | 2 | — |