Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CHFUZHKHPUYRJZ
|
8.5 | IC50 | 4 | — | |
IONVXRPWTRMITM
|
8.5 | Ki | 6 | — | |
MHIHRICEWVAMHY
|
8.5 | IC50 | 4 | — | |
UMMZZOSIEGYDTO
|
8.5 | Kd | 2 | — | |
DZCUBLTYHLRLAF
|
8.5 | IC50 | 2 | Yes | |
GNIYUURCQFKRCB
|
8.5 | IC50 | 11 | Yes | |
IGMQBINYIPIDJQ
|
8.5 | IC50 | 9 | Yes | |
MCIJHEGABQVOTC
|
8.5 | IC50 | 2 | — | |
SQQOETQMUXTTJU
|
8.5 | IC50 | 3 | — | |
GJYUDCNOWIRHBL
|
8.5 | IC50 | 5 | Yes | |
IPPGXRJXMXVNLN
|
8.5 | IC50 | 3 | — | |
KEFBHUKKKFYQSI
|
8.5 | IC50 | 2 | — | |
UUDQJODJTHYBOX
|
8.5 | IC50 | 2 | — | |
XXMJXRZJNGKMJK
|
8.5 | IC50 | 2 | — | |
YBXDKOSIYONZOF
|
8.5 | IC50 | 2 | — | |
DSRUNANRDDLTEB
|
8.5 | IC50 | 9 | — | |
GSFCLBKGTQCVGV
|
8.5 | IC50 | 2 | — | |
HGJSLQXBCKJGHL
|
8.5 | IC50 | 2 | — | |
KADQEUOYNAPXRD
|
8.5 | IC50 | 3 | Yes | |
LYADGAGFYYXXIO
|
8.5 | IC50 | 82 | — | |
PUHMCRONAFLMFJ
|
8.5 | IC50 | 2 | — | |
ZZOUIAPNOGIDSZ
|
8.5 | IC50 | 2 | Yes | |
BYRLMZPLBVGQSG
|
8.4 | IC50 | 2 | — | |
FNVQWCIBCILNCW
|
8.4 | Ki | 2 | — | |
HZORURMFPRFGNI
|
8.4 | IC50 | 2 | — | |
JLSKHZFXEMMJPA
|
8.4 | IC50 | 2 | — | |
LHKUVOGMYOGQMG
|
8.4 | Ki | 6 | — | |
SSMFYNNDUCDQGD
|
8.4 | IC50 | 2 | — | |
FKFACVZGGDYEHZ
|
8.4 | IC50 | 5 | Yes | |
GVVAOKGDOGVPSI
|
8.4 | IC50 | 2 | — | |
HZSSTZXPAUWYIN
|
8.4 | IC50 | 2 | — | |
JOJVJYUHAXMDPF
|
8.4 | IC50 | 2 | — | |
PKVCAQKGXZUIDA
|
8.4 | IC50 | 2 | — | |
VEVUBFZLKUNGER
|
8.4 | IC50 | 5 | — | |
WFMSTKDUQUETMD
|
8.4 | IC50 | 5 | — | |
BPCWWXWVIUQJOJ
|
8.4 | IC50 | 2 | — | |
FHTTVJXLZSYAJH
|
8.4 | Ki | 6 | — | |
FPZFOTHNFGTZRK
|
8.4 | IC50 | 2 | — | |
GCDSDVNITVBCDW
|
8.4 | IC50 | 17 | — | |
IKVZCSGUEDRZOZ
|
8.4 | IC50 | 2 | — | |
KBUOUGKAAPDJRZ
|
8.4 | IC50 | 2 | — | |
VSLNXMYUGRCLGS
|
8.4 | IC50 | 2 | — | |
VWWWKWXBDHJDSL
|
8.4 | IC50 | 2 | — | |
CPMDPSXJELVGJG
|
8.4 | Ki | 6 | — | |
HFLGPAUKVFOIOT
|
8.4 | IC50 | 4 | Yes | |
JEGKVDSRNBUXAN
|
8.4 | IC50 | 3 | — | |
NSKYYUZMAXEZIR
|
8.4 | Ki | 15 | — | |
POKUGRIXYDIRKM
|
8.4 | IC50 | 3 | — | |
RBZINWUMPZNWCZ
|
8.4 | IC50 | 4 | Yes | |
HUJRSGGBAXUNTD
|
8.4 | IC50 | 2 | — |