Target Details
| UniProt AC | P35968 |
|---|---|
| Gene Symbol | KDR |
| Protein Name | Vascular endothelial growth factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF13895 (Ig_2) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 5,667
- Clinical molecules 877
- Avg pChEMBL 7.23
KEGG Pathways (13)
- Cadherin signaling
- Calcium signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- IgSF CAM signaling
- Integrin signaling
- MAPK signaling pathway
- PI3K-Akt signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- VEGF signaling pathway
Associated Diseases (1)
Active Molecules (5,667)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WQIVPDKBAHQPEF
|
10.6 | IC50 | 2 | — | |
AMZNBJDLFWYTNW
|
10.5 | Ki | 2 | — | |
ITLTXJASMJITNS
|
10.5 | Ki | 2 | — | |
ONIQOQHATWINJY
|
10.5 | IC50 | 25 | — | |
JXSVVZKPEDIRTN
|
10.4 | Ki | 2 | — | |
UMNQEFXKDFGFNN
|
10.3 | Ki | 3 | — | |
BTYKIQPZILZZIK
|
10.2 | Ki | 2 | — | |
HPTVZCOLBBFDMI
|
10.0 | IC50 | 3 | — | |
KKJCDJULBOTJNL
|
10.0 | Ki | 2 | — | |
PGOFCHZWKNKRQH
|
9.8 | Ki | 2 | — | |
XPVAPOBXNPDLHJ
|
9.7 | IC50 | 3 | — | |
CJPNTWIJDMEPOG
|
9.7 | IC50 | 2 | — | |
DRBIGHXBYOJZLO
|
9.7 | IC50 | 3 | — | |
JGRUAZVMJJCPHI
|
9.7 | IC50 | 2 | — | |
JPTQVDRPKXSDDN
|
9.7 | IC50 | 3 | — | |
KSMZEXLVHXZPEF
|
9.7 | IC50 | 2 | — | |
URESLPMFUBHALD
|
9.7 | IC50 | 2 | — | |
YULUVWHIOGBTPX
|
9.7 | IC50 | 4 | Yes | |
RITAVMQDGBJQJZ
|
9.7 | IC50 | 43 | — | |
QIZGCINCAAEMBX
|
9.6 | IC50 | 2 | — | |
NKKLZQAIJJQHIF
|
9.6 | IC50 | 3 | — | |
SXKJHBJVKCAXFA
|
9.6 | IC50 | 3 | — | |
APJYLVNVUZIPJQ
|
9.6 | IC50 | 2 | — | |
JVVXCTKZKBXESA
|
9.5 | IC50 | 2 | — | |
ZPOKSLXILOTPCR
|
9.5 | IC50 | 2 | — | |
UMGGFVAOWVEZEZ
|
9.5 | IC50 | 3 | — | |
RFHIMTLASCGOTR
|
9.5 | IC50 | 3 | — | |
XKNVITFCGXBPNA
|
9.5 | IC50 | 2 | — | |
ZCSZQHZLTLCNBJ
|
9.5 | IC50 | 2 | — | |
MZZIULFUXGVMGF
|
9.5 | IC50 | 3 | — | |
BALLNEJQLSTPIO
|
9.5 | IC50 | 3 | — | |
LKWJIINNTXDWNN
|
9.4 | IC50 | 3 | — | |
LOCPAEPNEIAJSG
|
9.4 | IC50 | 2 | — | |
IAYJLHOAEWIYAY
|
9.4 | IC50 | 4 | Yes | |
MGMPLTIIDFSKQV
|
9.4 | Ki | 2 | — | |
ZDFUUQNEPJWJNC
|
9.4 | IC50 | 2 | — | |
DPRXHQKZIFLCDL
|
9.4 | IC50 | 2 | — | |
HOOKXRVARVUTOQ
|
9.4 | IC50 | 2 | — | |
NVMDAZMLLHNPND
|
9.4 | IC50 | 2 | — | |
BVSYMJUCSKOBAS
|
9.4 | IC50 | 2 | — | |
GCTNXTNPSNLYBZ
|
9.4 | IC50 | 4 | — | |
LBAQJHGPPPQHFJ
|
9.4 | IC50 | 2 | — | |
RJPGJHLVEUSRRA
|
9.4 | Ki | 2 | — | |
WTMJVPWFPQDGDL
|
9.4 | IC50 | 2 | — | |
OMASESMZSSNIBS
|
9.4 | IC50 | 2 | — | |
YFBBPYBKOLENKT
|
9.4 | IC50 | 2 | — | |
APJYLVNVUZIPJQ
|
9.4 | IC50 | 2 | — | |
IUZQUGLOCXBWCX
|
9.4 | IC50 | 2 | — | |
IFOVLFYNYABOTP
|
9.4 | IC50 | 2 | — | |
LYKFUIDYYBNHOA
|
9.4 | IC50 | 2 | — |