Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PEGWVOKOYYAQEV
|
6.9 | IC50 | 9 | — | |
GZOYOEIHAGHGFM
|
6.9 | IC50 | 6 | — | |
BHSOPYVVEZFHDB
|
6.9 | Ki | 25 | Yes | |
MADCXGNPDBWPLM
|
6.9 | Ki | 25 | — | |
NLUPJKQOKWBWFC
|
6.9 | Ki | 69 | — | |
TVJQMNOHJPUFKJ
|
6.9 | IC50 | 3 | — | |
VPBYZLCHOKSGRX
|
6.9 | IC50 | 4 | — | |
VRHNKAXZHXPLGK
|
6.9 | IC50 | 3 | — | |
VWVYILCFSYNJHF
|
6.9 | Ki | 49 | — | |
XYXLUJQBBIBJFV
|
6.9 | Ki | 36 | — | |
YACXOXQTGJXYNX
|
6.9 | Ki | 11 | — | |
XYFGHOWVIROTAV
|
6.9 | IC50 | 5 | Yes | |
GJIVVHLMOZQKEB
|
6.8 | IC50 | 3 | — | |
SKDBXDGKLQALIZ
|
6.8 | IC50 | 15 | — | |
ZIJIMHMKDXTURQ
|
6.8 | IC50 | 6 | Yes | |
RAOCKIXJWYDYCO
|
6.8 | IC50 | 5 | Yes | |
FAGREBOKSNRJQA
|
6.8 | IC50 | 3 | — | |
RFSFIDGEFVXSQM
|
6.8 | IC50 | 12 | Yes | |
ZBCIUJVPXUPSFS
|
6.8 | IC50 | 3 | — | |
AYJBHLUSGLQYDG
|
6.8 | Ki | 16 | — | |
HEUSUIRCBWROMH
|
6.8 | Ki | 64 | — | |
JSDGKSMNPHJDFK
|
6.8 | Ki | 35 | — | |
MOSKATHMXWSZTQ
|
6.8 | IC50 | 16 | Yes | |
OLUKILHGKRVDCT
|
6.8 | Ki | 44 | Yes | |
RAPYFGJGASETOS
|
6.8 | Ki | 11 | — | |
WUWDLXZGHZSWQZ
|
6.8 | IC50 | 11 | Yes | |
XKFTZKGMDDZMJI
|
6.8 | Ki | 56 | — | |
XLFYOIVELARSKP
|
6.8 | Ki | 33 | — | |
XKFTZKGMDDZMJI
|
6.8 | IC50 | 64 | Yes | |
AQFXVMZZFFFSCG
|
6.8 | IC50 | 5 | — | |
DHKRVOSGULPXFM
|
6.8 | IC50 | 3 | — | |
PQZKVWILKSYPCO
|
6.8 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
UNYBBLITYOSZKC
|
6.8 | IC50 | 2 | — | |
WWSUCZQRKHASNA
|
6.8 | IC50 | 3 | — | |
OODPPJDFRMJIDK
|
6.8 | IC50 | 3 | — | |
UZYXETLFKQALDE
|
6.8 | IC50 | 3 | — | |
LODWOBAYUQRWKD
|
6.7 | IC50 | 7 | — | |
DXCUKNQANPLTEJ
|
6.7 | IC50 | 7 | — | |
REIUSODTVBSVPQ
|
6.7 | IC50 | 3 | — | |
RGGYJEYZTPRESN
|
6.7 | IC50 | 6 | Yes | |
SDTAEHMYBHWTDK
|
6.7 | IC50 | 8 | Yes | |
YCOYDOIWSSHVCK
|
6.7 | Kd | 10 | — | |
AGYRJOAGMDIFKL
|
6.7 | Ki | 17 | — | |
AZJXTFAKHUFRQY
|
6.7 | IC50 | 3 | — | |
FUMCKNCUEAQHCV
|
6.7 | Ki | 103 | — | |
HAYYBYPASCDWEQ
|
6.7 | Ki | 47 | — | |
HTZZYCNEQVCJJB
|
6.7 | IC50 | 5 | Yes | |
LCGSWTFWYNYUKS
|
6.7 | Ki | 26 | — | |
NRSGWEVTVGZDFC
|
6.7 | Ki | 50 | — |