Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RAMCMRRBGWIDLK
|
7.2 | IC50 | 8 | Yes | |
QKPLUKMJEKRAJD
|
7.2 | IC50 | 30 | Yes | |
XMUWGNAFKPBEAU
|
7.2 | IC50 | 5 | Yes | |
OZWMSXPIQVMFDE
|
7.2 | IC50 | 8 | Yes | |
PBESGEKOQIKSKI
|
7.2 | IC50 | 5 | Yes | |
SCUGTCMSRMQNNQ
|
7.2 | IC50 | 7 | — | |
VEOIWTSZBRXBQG
|
7.2 | IC50 | 5 | Yes | |
NWEIPABWNQPRCZ
|
7.2 | IC50 | 7 | Yes | |
ABQSJCCISLWTEW
|
7.1 | IC50 | 8 | Yes | |
LSJAPABXQBDHRE
|
7.1 | IC50 | 5 | — | |
QXWNDTWKOGDJMG
|
7.1 | IC50 | 5 | — | |
UEJXELMBDCXXAQ
|
7.1 | IC50 | 9 | — | |
QTBWCSQGBMPECM
|
7.1 | IC50 | 21 | Yes | |
JGEBLDKNWBUGRZ
|
7.1 | IC50 | 20 | Yes | |
OSVUGUHRKMMBSE
|
7.1 | Kd | 170 | — | |
CQBBMNXXVMOFCA
|
7.1 | Ki | 39 | — | |
CXBBWVXSZINRCS
|
7.1 | Ki | 41 | — | |
LVECPYVAIBNSRV
|
7.1 | Ki | 33 | — | |
OZVUSEVFXCWUBV
|
7.1 | IC50 | 5 | Yes | |
SRUYMJRFVGLQDV
|
7.1 | Ki | 37 | — | |
ZXLFIHLBHMLHFJ
|
7.1 | Ki | 31 | — | |
YEIRROBVFZDCIW
|
7.1 | IC50 | 7 | — | |
GXKSGTIXGWDSGJ
|
7.1 | IC50 | 12 | Yes | |
LDRYCDRIKRFDRD
|
7.1 | IC50 | 5 | Yes | |
RGQCKSICTLMEDR
|
7.1 | IC50 | 3 | — | |
CPQMLGLUULWKDX
|
7.0 | IC50 | 4 | Yes | |
MMHADELJVDMSNQ
|
7.0 | IC50 | 7 | Yes | |
PGLZJHICUYCCJE
|
7.0 | IC50 | 7 | — | |
JSKUWFIZUALZLX
|
7.0 | IC50 | 33 | — | |
FYZOPODRENDNJN
|
7.0 | IC50 | 5 | Yes | |
GSFNVLNOUTVLFC
|
7.0 | IC50 | 5 | Yes | |
GWJHMRBQEUHFOC
|
7.0 | Ki | 42 | — | |
GXFGHUNNGNQSMQ
|
7.0 | Ki | 19 | — | |
ITQSJZWWFWDOKJ
|
7.0 | IC50 | 5 | Yes | |
JAMDNXUAYUHJLJ
|
7.0 | Ki | 40 | — | |
KIWKXIDEBINNAK
|
7.0 | IC50 | 5 | Yes | |
PKCDDUHJAFVJJB
|
7.0 | Ki | 13 | — | |
SEVCBWKJSOLMNQ
|
7.0 | Ki | 38 | — | |
XNEPVLVYFUGJLF
|
7.0 | Ki | 27 | — | |
ZWVZORIKUNOTCS
|
7.0 | Ki | 69 | — | |
DEXMHPPNXPZZKY
|
7.0 | IC50 | 3 | — | |
ZHLODYGHLUYMDJ
|
7.0 | IC50 | 7 | — | |
PKUDAUZYOFHVDW
|
7.0 | IC50 | 3 | — | |
ZYZUOYYVHYGMDE
|
7.0 | IC50 | 4 | — | |
PSNSRJNHZPJVJH
|
7.0 | IC50 | 18 | — | |
DGRCFAYRKDYEMX
|
6.9 | IC50 | 7 | — | |
QPIFMCLNACVAAT
|
6.9 | IC50 | 7 | — | |
CVMUHXWSBHMVGZ
|
6.9 | IC50 | 6 | Yes | |
DXQBCGUEDOHNHP
|
6.9 | Kd | 12 | — | |
ODPGGGTTYSGTGO
|
6.9 | Kd | 153 | — |