Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JAYZLGOACZERIJ
|
7.3 | IC50 | 7 | Yes | |
MJTPRNMULDHJJJ
|
7.3 | IC50 | 4 | — | |
PYUIBNGQBBAKFO
|
7.3 | IC50 | 7 | Yes | |
GUDCGYXTFRTWMP
|
7.3 | IC50 | 3 | — | |
LAJAFFLJAJMYLK
|
7.3 | IC50 | 17 | — | |
UXWPGZNWYZLVFJ
|
7.3 | IC50 | 3 | — | |
KBLQLKPQLQTCDT
|
7.3 | IC50 | 3 | — | |
BOBGABAXWFYHQX
|
7.3 | Ki | 9 | — | |
CKVWQORGCCEYHS
|
7.3 | Ki | 50 | — | |
CNTCGRJDUJEUDG
|
7.3 | Ki | 37 | — | |
CTNPALGJUAXMMC
|
7.3 | Kd | 151 | — | |
IOYGAWXBNPFOKF
|
7.3 | IC50 | 3 | — | |
JNAHSSCHKKAPHI
|
7.3 | IC50 | 5 | Yes | |
KNAJKXGUAHBQTI
|
7.3 | IC50 | 5 | Yes | |
KPPYNHRMNFKBRA
|
7.3 | IC50 | 7 | — | |
LSHMOEOLVFEUHJ
|
7.3 | IC50 | 5 | Yes | |
NWAUBAGBGOPJLF
|
7.3 | Ki | 51 | Yes | |
RKKIDHHGKNGTQI
|
7.3 | Ki | 28 | — | |
RTDSHUGNRVXRHN
|
7.3 | Ki | 51 | — | |
VDHBAAXTLJWVLI
|
7.3 | IC50 | 4 | Yes | |
YBTGTVGEKMZEQX
|
7.3 | IC50 | 5 | Yes | |
ZKHDDJKHTPLPOQ
|
7.3 | Ki | 62 | — | |
NGBFROQDGZCMCE
|
7.3 | IC50 | 3 | — | |
IGMQBINYIPIDJQ
|
7.3 | IC50 | 9 | Yes | |
GVEYCTQROBIZHZ
|
7.3 | IC50 | 5 | — | |
HXHAJRMTJXHJJZ
|
7.3 | IC50 | 52 | Yes | |
JKDOLJKPWNOURO
|
7.3 | IC50 | 3 | — | |
WCWUXEGQKLTGDX
|
7.2 | Kd | 22 | Yes | |
AILRADAXUVEEIR
|
7.2 | IC50 | 75 | — | |
NZTCZQRXCIAJMP
|
7.2 | IC50 | 5 | Yes | |
WIXHYLINPBKNTE
|
7.2 | IC50 | 5 | Yes | |
YOBIWCLAYQWPPW
|
7.2 | IC50 | 23 | — | |
ZMYSTIZWTSDYEP
|
7.2 | IC50 | 5 | — | |
AVQNSHZBOYOSQZ
|
7.2 | IC50 | 5 | Yes | |
JFGLOXKNWPNMQT
|
7.2 | IC50 | 5 | Yes | |
KQEHWOWUWGAOSR
|
7.2 | IC50 | 5 | Yes | |
OORQGKRPXSYBAR
|
7.2 | IC50 | 5 | Yes | |
LMHPBVGQEGWFGF
|
7.2 | IC50 | 3 | — | |
NXSJMRCTGYTSTK
|
7.2 | Kd | 200 | — | |
KKYPRNBBPBRJQX
|
7.2 | Ki | 40 | — | |
KYHMOCUKKUVQSG
|
7.2 | Ki | 3 | — | |
OUJZYQBEFNDJQN
|
7.2 | Ki | 71 | — | |
UDFDIIVNIYWXDM
|
7.2 | Ki | 74 | — | |
UWDBNTXEKYRMSG
|
7.2 | Ki | 26 | — | |
XSRHBCYNCKAFKS
|
7.2 | Ki | 45 | — | |
FZBVNCFBCNXULH
|
7.2 | IC50 | 18 | — | |
WPCUQWCGLJALCN
|
7.2 | IC50 | 4 | — | |
XKZQZMSAWVDRSP
|
7.2 | IC50 | 39 | Yes | |
HRUYZDJOLIPWLW
|
7.2 | IC50 | 5 | Yes | |
LQAMNACDVZLTDL
|
7.2 | IC50 | 5 | — |