Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OOQJIJYKWXLQNC
|
7.5 | IC50 | 16 | Yes | |
OSEYUXXMDLYZKE
|
7.5 | IC50 | 5 | Yes | |
VTWWRKFUHCSCEW
|
7.5 | Kd | 19 | — | |
FDVSOQRNTAPCHB
|
7.5 | Ki | 40 | — | |
GWMATETWMAQOFL
|
7.5 | Ki | 36 | — | |
NFKMFNBKEOQNPZ
|
7.5 | Ki | 43 | — | |
NFMGZVPRGVERNN
|
7.5 | Ki | 44 | — | |
PJYLAPUQQYSUKA
|
7.5 | IC50 | 5 | — | |
QJIVDCJIPGAKQZ
|
7.5 | Ki | 25 | — | |
SKZQZGSPYYHTQG
|
7.5 | IC50 | 3 | — | |
WVPSKSLAZQPAKQ
|
7.5 | Ki | 3 | — | |
ICESXCDRPZKRHM
|
7.5 | IC50 | 5 | — | |
GJYUDCNOWIRHBL
|
7.5 | IC50 | 5 | Yes | |
LDYBJNSNFYSDIW
|
7.5 | IC50 | 4 | Yes | |
BALLNEJQLSTPIO
|
7.5 | IC50 | 3 | — | |
JLXBHBVYBGZIEY
|
7.5 | IC50 | 7 | Yes | |
WDDLXDTWOAENKE
|
7.5 | IC50 | 5 | Yes | |
WINHZLLDWRZWRT
|
7.5 | Kd | 201 | Yes | |
MLDQJTXFUGDVEO
|
7.4 | IC50 | 85 | Yes | |
DSRUNANRDDLTEB
|
7.4 | IC50 | 9 | — | |
QNIMLRHYPMIYSE
|
7.4 | IC50 | 7 | Yes | |
QTIHZRQNFPNCHT
|
7.4 | IC50 | 4 | — | |
YTFRDKYCZHOSMM
|
7.4 | IC50 | 4 | Yes | |
RJUAJPXDDBGVQP
|
7.4 | IC50 | 2 | — | |
DYSDUQPAIATDAA
|
7.4 | IC50 | 5 | Yes | |
MAQBPYJYNOISMO
|
7.4 | IC50 | 4 | Yes | |
SCMLRESZJCKCTC
|
7.4 | IC50 | 7 | — | |
BMEKKWWFQMYXPU
|
7.4 | IC50 | 5 | Yes | |
DOKIBWCVABZHOH
|
7.4 | IC50 | 3 | — | |
JFGLOXKNWPNMQT
|
7.4 | IC50 | 4 | — | |
MULNSLQVKKUPJN
|
7.4 | Ki | 41 | — | |
QHXBWJSQXSYAGG
|
7.4 | IC50 | 16 | — | |
RWEHAHIEUDLKGT
|
7.4 | Ki | 33 | — | |
SPMHGQZFMNZCBV
|
7.4 | Ki | 30 | Yes | |
SWIHGAFGYUTAOY
|
7.4 | IC50 | 4 | — | |
ZDUNROKMXDSWQP
|
7.4 | IC50 | 4 | Yes | |
ZESRALQQFCOMOY
|
7.4 | IC50 | 5 | Yes | |
ZVWRFVCNQOECJS
|
7.4 | Ki | 71 | — | |
CVWXJKQAOSCOAB
|
7.4 | Kd | 35 | — | |
DEEQWPIMFASFIP
|
7.4 | IC50 | 7 | Yes | |
DYIBUWLFYBFBBS
|
7.4 | IC50 | 5 | — | |
FNHKPVJBJVTLMP
|
7.4 | IC50 | 29 | — | |
RWCSLXSUPQHKBX
|
7.4 | IC50 | 4 | Yes | |
JWILUIVAYLRFIY
|
7.4 | IC50 | 14 | — | |
YMKCMNJQFGEWCA
|
7.4 | IC50 | 8 | Yes | |
IXIJKXSIADDKHR
|
7.3 | IC50 | 12 | — | |
ZHOXAGNPCZTRBN
|
7.3 | Kd | 20 | — | |
CUIHSIWYWATEQL
|
7.3 | IC50 | 61 | Yes | |
IPBGKKBBYNOXCG
|
7.3 | IC50 | 10 | — | |
XYGDYCMPYIUPHS
|
7.3 | IC50 | 4 | Yes |