Target Details
| UniProt AC | P35916 |
|---|---|
| Gene Symbol | FLT4 |
| Protein Name | Vascular endothelial growth factor receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF13927 (Ig_3) PF22971 (Ig_VEGFR-1-like_5th) PF07714 (PK_Tyr_Ser-Thr) PF21339 (VEGFR-1-like_Ig-like) PF17988 (VEGFR-2_TMD) PF22854 (VEGFR1-3_N_Ig-like) |
Summary
- Multi-target molecules 636
- Clinical molecules 169
- Avg pChEMBL 7.35
KEGG Pathways (10)
Associated Diseases (4)
Active Molecules (636)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NZBQAOCZTUIYGZ
|
7.7 | IC50 | 3 | — | |
ORWIYCURPDKSBI
|
7.7 | IC50 | 15 | Yes | |
QBRQTJMZEYORSP
|
7.7 | Kd | 12 | — | |
RJUAJPXDDBGVQP
|
7.7 | IC50 | 2 | — | |
VTSUXBCLYFIJIZ
|
7.7 | IC50 | 2 | — | |
APPXQUDJLJXULP
|
7.7 | IC50 | 47 | — | |
DKSNLQYRZJKYOC
|
7.7 | Ki | 51 | — | |
FLEAYYMORDPWAJ
|
7.7 | Ki | 90 | — | |
RITAVMQDGBJQJZ
|
7.7 | Ki | 33 | — | |
SAZIXFAROZCPDO
|
7.7 | IC50 | 7 | Yes | |
YABJJWZLRMPFSI
|
7.7 | IC50 | 34 | — | |
AQXIMVWUURMKKC
|
7.7 | IC50 | 7 | Yes | |
FUTJVLYPEWQFEG
|
7.7 | IC50 | 2 | — | |
BFAFTEXTXVWPSX
|
7.7 | IC50 | 5 | Yes | |
MHHCPQUFBADOGH
|
7.7 | IC50 | 3 | — | |
OEZUXIBNCYTQAV
|
7.7 | IC50 | 5 | Yes | |
YUAOWJBCURIMGN
|
7.7 | IC50 | 3 | — | |
AMQUNUQXLQUCGJ
|
7.6 | IC50 | 3 | — | |
CBCKPZZVJQHROG
|
7.6 | IC50 | 5 | — | |
PVNVVSOCNKJUKM
|
7.6 | IC50 | 3 | — | |
VEVUBFZLKUNGER
|
7.6 | IC50 | 3 | — | |
GVZZEKBXTZEWOA
|
7.6 | IC50 | 2 | — | |
HFSWCNDZVPIIOF
|
7.6 | IC50 | 8 | — | |
HPTYEEJJIBEOEW
|
7.6 | IC50 | 5 | — | |
MJBOSKJANLJEQK
|
7.6 | IC50 | 5 | Yes | |
WMWHVTDZNIVNIE
|
7.6 | IC50 | 9 | — | |
WMWHVTDZNIVNIE
|
7.6 | IC50 | 9 | — | |
AIQDZMUPVYDVLB
|
7.6 | Ki | 48 | — | |
BSFNGHCTZDCQBF
|
7.6 | Ki | 93 | — | |
FWRUVEHMIVRQGU
|
7.6 | IC50 | 2 | — | |
KNCMFVBGBJGBGI
|
7.6 | IC50 | 7 | Yes | |
WINHZLLDWRZWRT
|
7.6 | Ki | 66 | — | |
PSWWUMTWJRPKLC
|
7.6 | IC50 | 3 | — | |
FAYFMVHYNQOQRQ
|
7.6 | IC50 | 7 | Yes | |
OIANGKGOYKDGQV
|
7.6 | Kd | 10 | — | |
RJUAJPXDDBGVQP
|
7.6 | IC50 | 2 | — | |
WAYBUMGYWVVITR
|
7.6 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
7.5 | Kd | 213 | — | |
PIQCTGMSNWUMAF
|
7.5 | IC50 | 137 | Yes | |
BJTVHTAPKJNNGR
|
7.5 | IC50 | 3 | — | |
CXMKJARIDJFGGI
|
7.5 | IC50 | 3 | — | |
FTDWSWREBGYXDZ
|
7.5 | IC50 | 10 | — | |
KRICMVKKVCDVBV
|
7.5 | IC50 | 7 | Yes | |
LDACHLNBCOVNBL
|
7.5 | IC50 | 8 | — | |
SIABKVPDKZOJCK
|
7.5 | IC50 | 5 | Yes | |
UVLOISNMRLZTPF
|
7.5 | IC50 | 5 | — | |
XLZFINWQTYEKJR
|
7.5 | IC50 | 5 | Yes | |
ZMAGOHAYMIZJEE
|
7.5 | IC50 | 5 | Yes | |
ZTHXTCUTPBRCGU
|
7.5 | IC50 | 5 | Yes | |
KULLGNXUHQGZIB
|
7.5 | IC50 | 3 | — |